| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 8.6 | 8.6 | 2.5 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Protein kinase C delta type CHEMBL2996 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| STE20-like serine/threonine-protein kinase CHEMBL4202 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Glycogen synthase kinase-3 beta CHEMBL262 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Tyrosine-protein kinase Fyn CHEMBL1841 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Ribosomal protein S6 kinase alpha-5 CHEMBL4237 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Casein kinase I isoform gamma-1 CHEMBL2426 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Casein kinase I isoform gamma-3 CHEMBL5084 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Cyclin-dependent kinase 7 CHEMBL3055 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Ribosomal protein S6 kinase beta-1 CHEMBL4501 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Proto-oncogene tyrosine-protein kinase Src CHEMBL267 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX CHEMBL5818 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Cyclin-dependent kinase 9 CHEMBL3116 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Macrophage colony-stimulating factor 1 receptor CHEMBL1844 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 6.7 | 6.7 | 199.5 | 1 |