Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1964116

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CSNK1G3
ChEMBL ↗
533
Total Activities
523
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Casein kinase I isoform gamma-3 (CHEMBL5084) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 533 5.96 8.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1999931 — — 1 8.10
CHEMBL1965660 — — 2 8.00
CHEMBL1969588 — — 1 7.70
CHEMBL2003638 — — 1 7.70
CHEMBL1990288 — — 2 7.50
CHEMBL1981079 — — 1 7.50
CHEMBL2006439 — — 1 7.50
CHEMBL1996066 — — 1 7.40
CHEMBL1966628 — — 1 7.30
CHEMBL1964290 — — 1 7.10
CHEMBL1998159 — — 1 7.10
CHEMBL1991078 — — 1 7.10
CHEMBL1989646 — — 1 7.00
CHEMBL1970903 — — 1 7.00
CHEMBL1994830 — — 1 7.00
CHEMBL1975900 — — 1 6.90
CHEMBL1982361 — — 1 6.90
CHEMBL1980489 — — 1 6.80
CHEMBL225519 — — 1 6.80
CHEMBL1978448 — — 1 6.80
CHEMBL1969843 — — 1 6.80
CHEMBL396523 — — 1 6.80
CHEMBL1991063 — — 1 6.80
CHEMBL1995813 — — 1 6.60
CHEMBL1971186 — — 1 6.60
CHEMBL1994864 — — 1 6.60
CHEMBL1974870 — — 1 6.60
CHEMBL243088 — — 1 6.60
CHEMBL1988173 — — 1 6.50
CHEMBL1986781 — — 1 6.50

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1999931 — Ki = 7.943 nM 8.10
CHEMBL1965660 — Ki = 10.0 nM 8.00
CHEMBL1965660 — Ki = 10.0 nM 8.00
CHEMBL2003638 — Ki = 19.95 nM 7.70
CHEMBL1969588 — Ki = 19.95 nM 7.70
CHEMBL1990288 — Ki = 31.62 nM 7.50
CHEMBL2006439 — Ki = 31.62 nM 7.50
CHEMBL1981079 — Ki = 31.62 nM 7.50
CHEMBL1996066 — Ki = 39.81 nM 7.40
CHEMBL1966628 — Ki = 50.12 nM 7.30
CHEMBL1998159 — Ki = 79.43 nM 7.10
CHEMBL1964290 — Ki = 79.43 nM 7.10
CHEMBL1991078 — Ki = 79.43 nM 7.10
CHEMBL1989646 — Ki = 100.0 nM 7.00
CHEMBL1970903 — Ki = 100.0 nM 7.00
CHEMBL1994830 — Ki = 100.0 nM 7.00
CHEMBL1982361 — Ki = 125.89 nM 6.90
CHEMBL1975900 — Ki = 125.89 nM 6.90
CHEMBL396523 — Ki = 158.49 nM 6.80
CHEMBL1991063 — Ki = 158.49 nM 6.80
CHEMBL1980489 — Ki = 158.49 nM 6.80
CHEMBL1978448 — Ki = 158.49 nM 6.80
CHEMBL1969843 — Ki = 158.49 nM 6.80
CHEMBL225519 — Ki = 158.49 nM 6.80
CHEMBL1990288 — Ki = 199.53 nM 6.70
CHEMBL1971186 — Ki = 251.19 nM 6.60
CHEMBL1995813 — Ki = 251.19 nM 6.60
CHEMBL243088 — Ki = 251.19 nM 6.60
CHEMBL1974870 — Ki = 251.19 nM 6.60
CHEMBL1994864 — Ki = 251.19 nM 6.60
CHEMBL1986781 — Ki = 316.23 nM 6.50
CHEMBL1988173 — Ki = 316.23 nM 6.50
CHEMBL244378 — Ki = 398.11 nM 6.40
CHEMBL1990885 — Ki = 501.19 nM 6.30
CHEMBL1988153 — Ki = 501.19 nM 6.30
CHEMBL1979252 — Ki = 501.19 nM 6.30
CHEMBL2005936 — Ki = 501.19 nM 6.30
CHEMBL1998414 — Ki = 501.19 nM 6.30
CHEMBL1972158 — Ki = 501.19 nM 6.30
CHEMBL1986186 — Ki = 501.19 nM 6.30
CHEMBL2002726 — Ki = 501.19 nM 6.30
CHEMBL1965836 — Ki = 501.19 nM 6.30
CHEMBL2000508 — Ki = 630.96 nM 6.20
CHEMBL2005899 — Ki = 630.96 nM 6.20
CHEMBL1986943 — Ki = 630.96 nM 6.20
CHEMBL1978014 — Ki = 630.96 nM 6.20
CHEMBL1986943 — Ki = 630.96 nM 6.20
CHEMBL1964692 — Ki = 630.96 nM 6.20
CHEMBL1682552 — Ki = 794.33 nM 6.10
CHEMBL1969301 — Ki = 794.33 nM 6.10