| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 9.3 | 9.3 | 0.5 | 1 |
| Cyclin-dependent kinase 8 CHEMBL5719 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Casein kinase I isoform gamma-3 CHEMBL5084 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Interleukin-1 receptor-associated kinase 1 CHEMBL3357 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Serine/threonine-protein kinase MRCK alpha CHEMBL4516 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Cyclin-dependent kinase 5 CHEMBL4036 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Casein kinase I isoform gamma-1 CHEMBL2426 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| NT-3 growth factor receptor CHEMBL5608 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Cyclin-dependent kinase 2 CHEMBL301 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 CHEMBL3587 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Vascular endothelial growth factor receptor 3 CHEMBL1955 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha CHEMBL4101 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Mitogen-activated protein kinase 1 CHEMBL4040 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Tyrosine-protein kinase Fer CHEMBL3982 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 CHEMBL1075115 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma CHEMBL3829 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Serine/threonine-protein kinase PLK1 CHEMBL3024 | Ki | 6.3 | 6.3 | 501.2 | 1 |
| Serine/threonine-protein kinase Sgk2 CHEMBL5794 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| cGMP-dependent protein kinase 1 CHEMBL4273 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Glycogen synthase kinase-3 alpha CHEMBL2850 | Ki | 6.1 | 6.1 | 794.3 | 1 |
| Serine/threonine-protein kinase 17A CHEMBL4525 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Protein kinase C gamma type CHEMBL2938 | Ki | 6.0 | 6.0 | 1000.0 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Mitogen-activated protein kinase 13 CHEMBL2939 | Ki | 5.9 | 5.9 | 1258.9 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta CHEMBL4121 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| Casein kinase I isoform alpha CHEMBL2793 | Ki | 5.8 | 5.8 | 1584.9 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 5.7 | 5.7 | 1995.3 | 1 |
| High affinity nerve growth factor receptor CHEMBL2815 | Ki | 5.7 | 5.7 | 1995.3 | 1 |