Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1963731

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CDC7
ChEMBL ↗
652
Total Activities
639
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cell division cycle 7-related protein kinase (CHEMBL5443) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 652 7.68 9.90

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1964519 — — 1 9.90
CHEMBL244793 — — 1 9.90
CHEMBL1986943 — — 2 9.80
CHEMBL2005509 — — 1 9.80
CHEMBL1965660 — — 2 9.70
CHEMBL1992220 — — 1 9.70
CHEMBL1980562 — — 1 9.60
CHEMBL1980253 — — 1 9.50
CHEMBL1996980 — — 1 9.50
CHEMBL1969151 — — 1 9.50
CHEMBL1973720 — — 2 9.50
CHEMBL1992363 — — 1 9.50
CHEMBL1982271 — — 1 9.50
CHEMBL1969221 — — 1 9.40
CHEMBL2005216 — — 1 9.40
CHEMBL1979933 — — 1 9.40
CHEMBL2002613 — — 1 9.40
CHEMBL1972339 — — 1 9.40
CHEMBL1981079 — — 1 9.40
CHEMBL2006450 — — 1 9.30
CHEMBL2006439 — — 1 9.30
CHEMBL1999931 — — 1 9.30
CHEMBL1967662 — — 1 9.20
CHEMBL1969473 — — 1 9.20
CHEMBL1987948 — — 1 9.20
CHEMBL2003638 — — 1 9.20
CHEMBL1980435 — — 1 9.10
CHEMBL1974870 — — 2 9.10
CHEMBL1980178 — — 1 9.10
CHEMBL1983595 — — 1 9.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1964519 — Ki = 0.1259 nM 9.90
CHEMBL244793 — Ki = 0.1259 nM 9.90
CHEMBL2005509 — Ki = 0.1585 nM 9.80
CHEMBL1986943 — Ki = 0.1585 nM 9.80
CHEMBL1986943 — Ki = 0.1585 nM 9.80
CHEMBL1965660 — Ki = 0.1995 nM 9.70
CHEMBL1992220 — Ki = 0.1995 nM 9.70
CHEMBL1965660 — Ki = 0.1995 nM 9.70
CHEMBL1980562 — Ki = 0.2512 nM 9.60
CHEMBL1992363 — Ki = 0.3162 nM 9.50
CHEMBL1982271 — Ki = 0.3162 nM 9.50
CHEMBL1996980 — Ki = 0.3162 nM 9.50
CHEMBL1980253 — Ki = 0.3162 nM 9.50
CHEMBL1973720 — Ki = 0.3162 nM 9.50
CHEMBL1969151 — Ki = 0.3162 nM 9.50
CHEMBL1973720 — Ki = 0.3162 nM 9.50
CHEMBL1979933 — Ki = 0.3981 nM 9.40
CHEMBL2002613 — Ki = 0.3981 nM 9.40
CHEMBL2005216 — Ki = 0.3981 nM 9.40
CHEMBL1981079 — Ki = 0.3981 nM 9.40
CHEMBL1972339 — Ki = 0.3981 nM 9.40
CHEMBL1969221 — Ki = 0.3981 nM 9.40
CHEMBL2006439 — Ki = 0.5012 nM 9.30
CHEMBL1999931 — Ki = 0.5012 nM 9.30
CHEMBL2006450 — Ki = 0.5012 nM 9.30
CHEMBL1967662 — Ki = 0.631 nM 9.20
CHEMBL2003638 — Ki = 0.631 nM 9.20
CHEMBL1987948 — Ki = 0.631 nM 9.20
CHEMBL1969473 — Ki = 0.631 nM 9.20
CHEMBL1980435 — Ki = 0.7943 nM 9.10
CHEMBL1974870 — Ki = 0.7943 nM 9.10
CHEMBL1980178 — Ki = 0.7943 nM 9.10
CHEMBL1974870 — Ki = 0.7943 nM 9.10
CHEMBL1996339 — Ki = 0.7943 nM 9.10
CHEMBL1983595 — Ki = 0.7943 nM 9.10
CHEMBL1966204 — Ki = 0.7943 nM 9.10
CHEMBL1998470 — Ki = 0.7943 nM 9.10
CHEMBL1970821 — Ki = 0.7943 nM 9.10
CHEMBL1968930 — Ki = 1.0 nM 9.00
CHEMBL2005718 — Ki = 1.0 nM 9.00
CHEMBL1998432 — Ki = 1.0 nM 9.00
CHEMBL385478 — Ki = 1.0 nM 9.00
CHEMBL2006456 — Ki = 1.0 nM 9.00
CHEMBL1971172 — Ki = 1.0 nM 9.00
CHEMBL1986855 — Ki = 1.0 nM 9.00
CHEMBL1991674 — Ki = 1.0 nM 9.00
CHEMBL1976936 — Ki = 1.0 nM 9.00
CHEMBL1999153 — Ki = 1.259 nM 8.90
CHEMBL1991078 — Ki = 1.259 nM 8.90
CHEMBL1988331 — Ki = 1.259 nM 8.90