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Assay Detail

CHEMBL1963783

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: CSNK1D
ChEMBL ↗
747
Total Activities
735
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Casein kinase I isoform delta (CHEMBL2828) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 747 6.16 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1990288 — — 2 8.30
CHEMBL2001547 — — 1 8.10
CHEMBL1994040 — — 1 8.10
CHEMBL1990904 — — 1 8.10
CHEMBL1986781 — — 1 8.10
CHEMBL1982383 — — 1 8.10
CHEMBL2000429 — — 1 8.00
CHEMBL1991800 — — 1 8.00
CHEMBL2000508 — — 1 8.00
CHEMBL2001957 — — 1 8.00
CHEMBL274064 SB-220025 — 1 7.90
CHEMBL1991678 — — 1 7.90
CHEMBL1995832 — — 1 7.90
CHEMBL1965660 — — 2 7.80
CHEMBL1987648 — — 1 7.80
CHEMBL1991395 — — 1 7.80
CHEMBL2005792 — — 1 7.80
CHEMBL1976093 — — 1 7.80
CHEMBL1984700 — — 1 7.80
CHEMBL1969372 — — 1 7.80
CHEMBL1986943 — — 2 7.70
CHEMBL1982563 — — 1 7.70
CHEMBL2000408 — — 1 7.70
CHEMBL95692 SB-242235 — 1 7.70
CHEMBL1966628 — — 1 7.60
CHEMBL363648 TAK-715 2.0 1 7.60
CHEMBL1981079 — — 1 7.60
CHEMBL1968127 — — 1 7.60
CHEMBL1965589 — — 1 7.60
CHEMBL256835 — — 1 7.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1990288 — Ki = 5.012 nM 8.30
CHEMBL1994040 — Ki = 7.943 nM 8.10
CHEMBL1986781 — Ki = 7.943 nM 8.10
CHEMBL1982383 — Ki = 7.943 nM 8.10
CHEMBL1990904 — Ki = 7.943 nM 8.10
CHEMBL2001547 — Ki = 7.943 nM 8.10
CHEMBL1991800 — Ki = 10.0 nM 8.00
CHEMBL2000508 — Ki = 10.0 nM 8.00
CHEMBL1990288 — Ki = 10.0 nM 8.00
CHEMBL2000429 — Ki = 10.0 nM 8.00
CHEMBL2001957 — Ki = 10.0 nM 8.00
CHEMBL1995832 — Ki = 12.59 nM 7.90
CHEMBL1991678 — Ki = 12.59 nM 7.90
CHEMBL274064 SB-220025 Ki = 12.59 nM 7.90
CHEMBL2005792 — Ki = 15.85 nM 7.80
CHEMBL1991395 — Ki = 15.85 nM 7.80
CHEMBL1987648 — Ki = 15.85 nM 7.80
CHEMBL1969372 — Ki = 15.85 nM 7.80
CHEMBL1984700 — Ki = 15.85 nM 7.80
CHEMBL1976093 — Ki = 15.85 nM 7.80
CHEMBL1965660 — Ki = 15.85 nM 7.80
CHEMBL1965660 — Ki = 15.85 nM 7.80
CHEMBL1986943 — Ki = 19.95 nM 7.70
CHEMBL1982563 — Ki = 19.95 nM 7.70
CHEMBL95692 SB-242235 Ki = 19.95 nM 7.70
CHEMBL1986943 — Ki = 19.95 nM 7.70
CHEMBL2000408 — Ki = 19.95 nM 7.70
CHEMBL17370 — Ki = 25.12 nM 7.60
CHEMBL1966628 — Ki = 25.12 nM 7.60
CHEMBL1981079 — Ki = 25.12 nM 7.60
CHEMBL256835 — Ki = 25.12 nM 7.60
CHEMBL1965589 — Ki = 25.12 nM 7.60
CHEMBL1968127 — Ki = 25.12 nM 7.60
CHEMBL1997617 — Ki = 25.12 nM 7.60
CHEMBL363648 TAK-715 Ki = 25.12 nM 7.60
CHEMBL1969735 — Ki = 31.62 nM 7.50
CHEMBL1974870 — Ki = 31.62 nM 7.50
CHEMBL1996500 — Ki = 31.62 nM 7.50
CHEMBL1984842 — Ki = 31.62 nM 7.50
CHEMBL1997129 — Ki = 31.62 nM 7.50
CHEMBL1725279 SP-600125 Ki = 31.62 nM 7.50
CHEMBL1978200 — Ki = 31.62 nM 7.50
CHEMBL504950 — Ki = 31.62 nM 7.50
CHEMBL10 SB-203580 Ki = 39.81 nM 7.40
CHEMBL1991063 — Ki = 39.81 nM 7.40
CHEMBL482967 CYC-116 Ki = 50.12 nM 7.30
CHEMBL1976090 — Ki = 50.12 nM 7.30
CHEMBL225519 — Ki = 50.12 nM 7.30
CHEMBL2003657 — Ki = 50.12 nM 7.30
CHEMBL2006439 — Ki = 63.1 nM 7.20