| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Casein kinase I isoform gamma-2 CHEMBL2543 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 CHEMBL5330 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Serine/threonine-protein kinase D2 CHEMBL4900 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase Chk2 CHEMBL2527 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Aurora kinase B CHEMBL2185 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Death-associated protein kinase 3 CHEMBL2468 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Dual specificity protein kinase CLK2 CHEMBL4225 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Casein kinase I isoform delta CHEMBL2828 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase N2 CHEMBL3032 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| Serine/threonine-protein kinase BRSK1 CHEMBL5650 | Ki | 7.4 | 7.4 | 39.8 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Tyrosine-protein kinase receptor UFO CHEMBL4895 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Casein kinase I isoform alpha CHEMBL2793 | Ki | 7.3 | 7.3 | 50.1 | 1 |
| Mitogen-activated protein kinase 8 CHEMBL2276 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Misshapen-like kinase 1 CHEMBL5518 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| MAP kinase-activated protein kinase 5 CHEMBL3094 | Ki | 7.2 | 7.2 | 63.1 | 1 |
| Serine/threonine-protein kinase MARK2 CHEMBL3831 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Mitogen-activated protein kinase 9 CHEMBL4179 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 7.1 | 7.1 | 79.4 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 7.0 | 7.0 | 100.0 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 CHEMBL4852 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha CHEMBL3476 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Mitogen-activated protein kinase 13 CHEMBL2939 | Ki | 6.9 | 6.9 | 125.9 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta CHEMBL1991 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform CHEMBL2349 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 | Ki | 6.8 | 6.8 | 158.5 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 6.7 | 6.7 | 199.5 | 1 |
| Mitogen-activated protein kinase 12 CHEMBL4674 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Serine/threonine-protein kinase pim-1 CHEMBL2147 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Homeodomain-interacting protein kinase 4 CHEMBL1075167 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Cyclin-dependent kinase 1 CHEMBL308 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Tyrosine-protein kinase Lck CHEMBL258 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Homeodomain-interacting protein kinase 2 CHEMBL4576 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 6.6 | 6.6 | 251.2 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| SRSF protein kinase 1 CHEMBL4375 | Ki | 6.5 | 6.5 | 316.2 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Epidermal growth factor receptor CHEMBL203 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Casein kinase II subunit alpha CHEMBL3629 | Ki | 6.4 | 6.4 | 398.1 | 1 |
| Maternal embryonic leucine zipper kinase CHEMBL4578 | Ki | 6.4 | 6.4 | 398.1 | 1 |