Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1963703

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: PRKCD
ChEMBL ↗
751
Total Activities
741
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category other
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Protein kinase C delta type (CHEMBL2996) ↗
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 751 5.94 8.50

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1966628 — — 1 8.50
CHEMBL220241 GSK-269962A — 1 8.30
CHEMBL1997534 — — 1 8.10
CHEMBL1969588 — — 1 8.10
CHEMBL2002726 — — 1 8.10
CHEMBL1965845 — — 1 8.00
CHEMBL2000271 — — 1 7.80
CHEMBL340384 — — 1 7.80
CHEMBL1990254 — — 2 7.80
CHEMBL2001751 — — 1 7.70
CHEMBL392642 — — 1 7.70
CHEMBL1976240 — — 1 7.60
CHEMBL1967887 — — 1 7.50
CHEMBL1970217 — — 1 7.40
CHEMBL1966524 — — 1 7.30
CHEMBL246970 — — 1 7.30
CHEMBL1986943 — — 2 7.20
CHEMBL1975121 — — 2 7.20
CHEMBL1991188 — — 1 7.20
CHEMBL1993661 — — 1 7.10
CHEMBL2006188 — — 1 7.00
CHEMBL1967878 CENISERTIB 2.0 1 7.00
CHEMBL1979554 — — 1 7.00
CHEMBL2004934 — — 1 6.90
CHEMBL1969049 — — 1 6.90
CHEMBL1974328 — — 1 6.90
CHEMBL1991674 — — 1 6.90
CHEMBL2002992 — — 1 6.80
CHEMBL1965660 — — 2 6.80
CHEMBL2000894 — — 1 6.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1966628 — Ki = 3.162 nM 8.50
CHEMBL220241 GSK-269962A Ki = 5.012 nM 8.30
CHEMBL1969588 — Ki = 7.943 nM 8.10
CHEMBL1997534 — Ki = 7.943 nM 8.10
CHEMBL2002726 — Ki = 7.943 nM 8.10
CHEMBL1965845 — Ki = 10.0 nM 8.00
CHEMBL1990254 — Ki = 15.85 nM 7.80
CHEMBL2000271 — Ki = 15.85 nM 7.80
CHEMBL340384 — Ki = 15.85 nM 7.80
CHEMBL1990254 — Ki = 15.85 nM 7.80
CHEMBL2001751 — Ki = 19.95 nM 7.70
CHEMBL392642 — Ki = 19.95 nM 7.70
CHEMBL1976240 — Ki = 25.12 nM 7.60
CHEMBL1967887 — Ki = 31.62 nM 7.50
CHEMBL1970217 — Ki = 39.81 nM 7.40
CHEMBL246970 — Ki = 50.12 nM 7.30
CHEMBL1966524 — Ki = 50.12 nM 7.30
CHEMBL1991188 — Ki = 63.1 nM 7.20
CHEMBL1975121 — Ki = 63.1 nM 7.20
CHEMBL1986943 — Ki = 63.1 nM 7.20
CHEMBL1986943 — Ki = 63.1 nM 7.20
CHEMBL1993661 — Ki = 79.43 nM 7.10
CHEMBL1979554 — Ki = 100.0 nM 7.00
CHEMBL1967878 CENISERTIB Ki = 100.0 nM 7.00
CHEMBL2006188 — Ki = 100.0 nM 7.00
CHEMBL1974328 — Ki = 125.89 nM 6.90
CHEMBL2004934 — Ki = 125.89 nM 6.90
CHEMBL1969049 — Ki = 125.89 nM 6.90
CHEMBL1991674 — Ki = 125.89 nM 6.90
CHEMBL1991180 — Ki = 158.49 nM 6.80
CHEMBL1969502 — Ki = 158.49 nM 6.80
CHEMBL2004771 — Ki = 158.49 nM 6.80
CHEMBL1965660 — Ki = 158.49 nM 6.80
CHEMBL2000894 — Ki = 158.49 nM 6.80
CHEMBL1965660 — Ki = 158.49 nM 6.80
CHEMBL2002992 — Ki = 158.49 nM 6.80
CHEMBL1967302 — Ki = 199.53 nM 6.70
CHEMBL1995813 — Ki = 199.53 nM 6.70
CHEMBL302449 GO-6976 Ki = 199.53 nM 6.70
CHEMBL1988608 — Ki = 199.53 nM 6.70
CHEMBL1987679 — Ki = 251.19 nM 6.60
CHEMBL1971029 — Ki = 251.19 nM 6.60
CHEMBL1999931 — Ki = 251.19 nM 6.60
CHEMBL340921 — Ki = 251.19 nM 6.60
CHEMBL1972158 — Ki = 251.19 nM 6.60
CHEMBL1987034 — Ki = 251.19 nM 6.60
CHEMBL1991728 — Ki = 316.23 nM 6.50
CHEMBL1993166 — Ki = 316.23 nM 6.50
CHEMBL592030 — Ki = 316.23 nM 6.50
CHEMBL1082440 — Ki = 316.23 nM 6.50