| Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 | Ki | 9.5 | 9.5 | 0.3 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 | Ki | 9.4 | 9.4 | 0.4 | 1 |
| MAP/microtubule affinity-regulating kinase 4 CHEMBL5754 | Ki | 9.3 | 9.3 | 0.5 | 1 |
| Mitogen-activated protein kinase kinase kinase 10 CHEMBL2873 | Ki | 9.1 | 9.1 | 0.8 | 1 |
| Tyrosine-protein kinase JAK2 CHEMBL2971 | Ki | 9.1 | 9.1 | 0.8 | 1 |
| Tyrosine-protein kinase Blk CHEMBL2250 | Ki | 9.0 | 9.0 | 1.0 | 1 |
| Tyrosine-protein kinase FRK CHEMBL4223 | Ki | 9.0 | 9.0 | 1.0 | 1 |
| Serine/threonine-protein kinase SIK2 CHEMBL5699 | Ki | 9.0 | 9.0 | 1.0 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 2 CHEMBL5284 | Ki | 8.9 | 8.9 | 1.3 | 1 |
| Fibroblast growth factor receptor 3 CHEMBL2742 | Ki | 8.8 | 8.8 | 1.6 | 1 |
| Serine/threonine-protein kinase PAK 4 CHEMBL4482 | Ki | 8.8 | 8.8 | 1.6 | 1 |
| Focal adhesion kinase 1 CHEMBL2695 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Tyrosine-protein kinase ITK/TSK CHEMBL2959 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Serine/threonine-protein kinase PLK4 CHEMBL3788 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Leukocyte tyrosine kinase receptor CHEMBL5627 | Ki | 8.5 | 8.5 | 3.2 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Interleukin-1 receptor-associated kinase 4 CHEMBL3778 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Mitogen-activated protein kinase 1 CHEMBL4040 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| ALK tyrosine kinase receptor CHEMBL4247 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Activated CDC42 kinase 1 CHEMBL4599 | Ki | 8.4 | 8.4 | 4.0 | 1 |
| Insulin-like growth factor 1 receptor CHEMBL1957 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Aurora kinase A CHEMBL4722 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Cell division cycle 7-related protein kinase CHEMBL5443 | Ki | 8.3 | 8.3 | 5.0 | 1 |
| Ephrin type-A receptor 2 CHEMBL2068 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Tyrosine-protein kinase JAK3 CHEMBL2148 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 CHEMBL3553 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 CHEMBL4045 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 | Ki | 8.2 | 8.2 | 6.3 | 1 |
| Tyrosine-protein kinase ABL1 CHEMBL1862 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Macrophage-stimulating protein receptor CHEMBL2689 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Testis-specific serine/threonine-protein kinase 1 CHEMBL6003 | Ki | 8.1 | 8.1 | 7.9 | 1 |
| Ribosomal protein S6 kinase alpha-3 CHEMBL2345 | Ki | 8.0 | 8.0 | 10.0 | 1 |
| Rho-associated protein kinase 1 CHEMBL3231 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Fibroblast growth factor receptor 1 CHEMBL3650 | Ki | 7.9 | 7.9 | 12.6 | 1 |
| Vascular endothelial growth factor receptor 2 CHEMBL279 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Serine/threonine-protein kinase Nek4 CHEMBL5819 | Ki | 7.8 | 7.8 | 15.8 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| LIM domain kinase 1 CHEMBL3836 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| BDNF/NT-3 growth factors receptor CHEMBL4898 | Ki | 7.7 | 7.7 | 19.9 | 1 |
| Vascular endothelial growth factor receptor 1 CHEMBL1868 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Mitogen-activated protein kinase 10 CHEMBL2637 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Rho-associated protein kinase 2 CHEMBL2973 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Dual specificity protein kinase CLK4 CHEMBL4203 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Serine/threonine-protein kinase TAO1 CHEMBL5261 | Ki | 7.6 | 7.6 | 25.1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Cyclin-dependent kinase 7 CHEMBL3055 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Hepatocyte growth factor receptor CHEMBL3717 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase PAK 1 CHEMBL4600 | Ki | 7.5 | 7.5 | 31.6 | 1 |
| Serine/threonine-protein kinase D3 CHEMBL2595 | Ki | 7.4 | 7.4 | 39.8 | 1 |