Assay Detail
Functional
CHEMBL1963740
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: FGFR1
1004
Total Activities
987
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1004 | 6.08 | 8.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2006778 | — | — | 1 | 8.80 |
| CHEMBL2005631 | — | — | 1 | 8.50 |
| CHEMBL1997924 | — | — | 1 | 8.30 |
| CHEMBL49120 | PD-0166285 | 1.0 | 1 | 8.30 |
| CHEMBL1989708 | — | — | 2 | 8.20 |
| CHEMBL1982476 | — | — | 1 | 8.20 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 8.10 |
| CHEMBL1984162 | — | — | 1 | 8.10 |
| CHEMBL1967116 | — | — | 1 | 8.10 |
| CHEMBL1987054 | — | — | 1 | 8.00 |
| CHEMBL1997617 | — | — | 1 | 8.00 |
| CHEMBL1969102 | — | — | 1 | 7.90 |
| CHEMBL1981047 | — | — | 1 | 7.90 |
| CHEMBL1979516 | — | — | 1 | 7.90 |
| CHEMBL1993661 | — | — | 1 | 7.90 |
| CHEMBL1973516 | — | — | 2 | 7.80 |
| CHEMBL253969 | OSI-632 | 2.0 | 1 | 7.80 |
| CHEMBL2000335 | — | — | 1 | 7.80 |
| CHEMBL1999414 | — | — | 1 | 7.80 |
| CHEMBL1970142 | — | — | 1 | 7.70 |
| CHEMBL1977148 | — | — | 1 | 7.70 |
| CHEMBL1998585 | — | — | 1 | 7.70 |
| CHEMBL1983111 | — | — | 1 | 7.70 |
| CHEMBL1972220 | — | — | 1 | 7.70 |
| CHEMBL1968590 | — | — | 1 | 7.70 |
| CHEMBL1970083 | — | — | 1 | 7.70 |
| CHEMBL1997822 | — | — | 1 | 7.70 |
| CHEMBL491473 | CEDIRANIB | 3.0 | 1 | 7.60 |
| CHEMBL1965988 | — | — | 1 | 7.60 |
| CHEMBL522892 | DOVITINIB | 3.0 | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2006778 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL2005631 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1997924 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL49120 | PD-0166285 | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1982476 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1989708 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1984162 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1989708 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1967116 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1997617 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1987054 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1993661 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1969102 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1981047 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1979516 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1973516 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL253969 | OSI-632 | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL2000335 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1999414 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1970142 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1983111 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1970083 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1972220 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1977148 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1997822 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1998585 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1968590 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1986851 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1971947 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL2007421 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1973540 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1981725 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1965988 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL371206 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1973516 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL509032 | TAE-684 | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL491473 | CEDIRANIB | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL522892 | DOVITINIB | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1974254 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1988387 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1994321 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2004716 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2002165 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1241473 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL262433 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL196363 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1967720 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1980995 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1988437 | — | Ki | = | 50.12 | nM | 7.30 |