Assay Detail
Functional
CHEMBL1963774
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: WEE1
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 34 | 7.44 | 9.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL379975 | — | — | 1 | 9.60 |
| CHEMBL49120 | PD-0166285 | 1.0 | 1 | 9.30 |
| CHEMBL1973516 | — | — | 1 | 8.60 |
| CHEMBL1967998 | — | — | 1 | 8.50 |
| CHEMBL1971914 | — | — | 1 | 8.10 |
| CHEMBL1999485 | — | — | 1 | 8.10 |
| CHEMBL1979690 | — | — | 1 | 8.10 |
| CHEMBL1974061 | — | — | 1 | 7.80 |
| CHEMBL1999484 | — | — | 1 | 7.10 |
| CHEMBL1242995 | — | — | 1 | 7.10 |
| CHEMBL1973961 | — | — | 1 | 7.10 |
| CHEMBL1988838 | — | — | 1 | 6.90 |
| CHEMBL1995703 | — | — | 1 | 6.90 |
| CHEMBL1983430 | — | — | 1 | 6.80 |
| CHEMBL1983715 | — | — | 1 | 6.70 |
| CHEMBL1083785 | — | — | 1 | 6.70 |
| CHEMBL482967 | CYC-116 | 1.0 | 1 | 6.30 |
| CHEMBL1968015 | — | — | 1 | 6.00 |
| CHEMBL1980995 | — | — | 1 | 5.70 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | - |
| CHEMBL1996048 | — | — | 1 | - |
| CHEMBL461876 | — | — | 1 | - |
| CHEMBL1980163 | — | — | 1 | - |
| CHEMBL1964648 | — | — | 1 | - |
| CHEMBL1983268 | ENTRECTINIB | 4.0 | 1 | - |
| CHEMBL1995201 | — | — | 1 | - |
| CHEMBL509032 | TAE-684 | — | 1 | - |
| CHEMBL1989043 | — | — | 1 | - |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | - |
| CHEMBL1825138 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL379975 | — | Ki | = | 0.2512 | nM | 9.60 |
| CHEMBL49120 | PD-0166285 | Ki | = | 0.5012 | nM | 9.30 |
| CHEMBL1973516 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL1967998 | — | Ki | = | 3.162 | nM | 8.50 |
| CHEMBL1971914 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1999485 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1979690 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1974061 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1999484 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1242995 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1973961 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL1988838 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL1995703 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL1983430 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL1083785 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1983715 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL482967 | CYC-116 | Ki | = | 501.19 | nM | 6.30 |
| CHEMBL1968015 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL1980995 | — | Ki | = | 1995.26 | nM | 5.70 |
| CHEMBL189963 | PALBOCICLIB | Ki | > | 3162.28 | nM | - |
| CHEMBL1996048 | — | Ki | > | 2511.89 | nM | - |
| CHEMBL461876 | — | Ki | > | 2511.89 | nM | - |
| CHEMBL1980163 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL1964648 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL1983268 | ENTRECTINIB | Ki | > | 2511.89 | nM | - |
| CHEMBL1995201 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL509032 | TAE-684 | Ki | > | 251.19 | nM | - |
| CHEMBL1989043 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL1967878 | CENISERTIB | Ki | > | 3162.28 | nM | - |
| CHEMBL1825138 | — | Ki | > | 2511.89 | nM | - |
| CHEMBL1164265 | — | Ki | > | 2511.89 | nM | - |
| CHEMBL1971556 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL1974582 | — | Ki | > | 3162.28 | nM | - |
| CHEMBL1230122 | R-1487 | Ki | > | 3162.28 | nM | - |