Assay Detail
Functional
CHEMBL1963732
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: RPS6KA4
32
Total Activities
32
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 32 | 6.77 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1987679 | — | — | 1 | 7.70 |
| CHEMBL2002726 | — | — | 1 | 7.40 |
| CHEMBL223360 | LINIFANIB | 3.0 | 1 | 7.30 |
| CHEMBL1990885 | — | — | 1 | 7.20 |
| CHEMBL1998585 | — | — | 1 | 7.10 |
| CHEMBL220057 | — | — | 1 | 7.00 |
| CHEMBL1964687 | — | — | 1 | 7.00 |
| CHEMBL2001257 | — | — | 1 | 6.90 |
| CHEMBL394619 | — | — | 1 | 6.80 |
| CHEMBL271381 | — | — | 1 | 6.80 |
| CHEMBL1973937 | — | — | 1 | 6.70 |
| CHEMBL1979883 | — | — | 1 | 6.70 |
| CHEMBL404367 | — | — | 1 | 6.60 |
| CHEMBL1973211 | — | — | 1 | 6.60 |
| CHEMBL1998545 | — | — | 1 | 6.20 |
| CHEMBL340921 | — | — | 1 | 6.10 |
| CHEMBL1991143 | — | — | 1 | 5.90 |
| CHEMBL1969755 | — | — | 1 | 5.80 |
| CHEMBL1975233 | — | — | 1 | - |
| CHEMBL387971 | — | — | 1 | - |
| CHEMBL941 | IMATINIB | 4.0 | 1 | - |
| CHEMBL1991285 | — | — | 1 | - |
| CHEMBL210887 | — | — | 1 | - |
| CHEMBL1992306 | — | — | 1 | - |
| CHEMBL10 | SB-203580 | — | 1 | - |
| CHEMBL2001224 | — | — | 1 | - |
| CHEMBL2006493 | — | — | 1 | - |
| CHEMBL253969 | OSI-632 | 2.0 | 1 | - |
| CHEMBL1973145 | — | — | 1 | - |
| CHEMBL402846 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1987679 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL2002726 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL223360 | LINIFANIB | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL1990885 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1998585 | — | Ki | = | 79.43 | nM | 7.10 |
| CHEMBL220057 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL1964687 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL2001257 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL394619 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL271381 | — | Ki | = | 158.49 | nM | 6.80 |
| CHEMBL1973937 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL1979883 | — | Ki | = | 199.53 | nM | 6.70 |
| CHEMBL404367 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1973211 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1998545 | — | Ki | = | 630.96 | nM | 6.20 |
| CHEMBL340921 | — | Ki | = | 794.33 | nM | 6.10 |
| CHEMBL1991143 | — | Ki | = | 1258.93 | nM | 5.90 |
| CHEMBL1969755 | — | Ki | = | 1584.89 | nM | 5.80 |
| CHEMBL1975233 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL387971 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL941 | IMATINIB | Ki | > | 1584.89 | nM | - |
| CHEMBL1991285 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL210887 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1992306 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL10 | SB-203580 | Ki | > | 1584.89 | nM | - |
| CHEMBL2001224 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL2006493 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL253969 | OSI-632 | Ki | > | 1584.89 | nM | - |
| CHEMBL1973145 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL402846 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL2004447 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL939 | GEFITINIB | Ki | > | 1584.89 | nM | - |