Assay Detail
Functional
CHEMBL1963810
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: MAP4K5
679
Total Activities
667
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Mitogen-activated protein kinase kinase kinase kinase 5 (CHEMBL4852) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 679 | 6.41 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1996649 | — | — | 1 | 9.70 |
| CHEMBL1999414 | — | — | 1 | 9.70 |
| CHEMBL1980995 | — | — | 1 | 9.20 |
| CHEMBL1979773 | — | — | 1 | 9.10 |
| CHEMBL1986851 | — | — | 1 | 8.90 |
| CHEMBL1970317 | — | — | 1 | 8.80 |
| CHEMBL1981725 | — | — | 1 | 8.40 |
| CHEMBL379975 | — | — | 1 | 8.40 |
| CHEMBL1966514 | — | — | 1 | 8.40 |
| CHEMBL1964692 | — | — | 1 | 8.30 |
| CHEMBL1994669 | — | — | 1 | 8.30 |
| CHEMBL1090360 | — | — | 1 | 8.30 |
| CHEMBL1981133 | — | — | 1 | 8.30 |
| CHEMBL1979883 | — | — | 1 | 8.20 |
| CHEMBL371206 | — | — | 1 | 8.20 |
| CHEMBL1965988 | — | — | 1 | 8.20 |
| CHEMBL508928 | — | — | 1 | 8.20 |
| CHEMBL1994321 | — | — | 1 | 8.10 |
| CHEMBL1973211 | — | — | 1 | 8.10 |
| CHEMBL49120 | PD-0166285 | 1.0 | 1 | 8.10 |
| CHEMBL1967531 | — | — | 1 | 8.10 |
| CHEMBL2005828 | — | — | 1 | 8.00 |
| CHEMBL1967878 | CENISERTIB | 2.0 | 1 | 8.00 |
| CHEMBL2006778 | — | — | 1 | 7.90 |
| CHEMBL1991429 | — | — | 1 | 7.90 |
| CHEMBL2006715 | — | — | 1 | 7.90 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.80 |
| CHEMBL1969190 | — | — | 1 | 7.80 |
| CHEMBL1982465 | — | — | 1 | 7.80 |
| CHEMBL1990885 | — | — | 1 | 7.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1996649 | — | Ki | = | 0.1995 | nM | 9.70 |
| CHEMBL1999414 | — | Ki | = | 0.1995 | nM | 9.70 |
| CHEMBL1980995 | — | Ki | = | 0.631 | nM | 9.20 |
| CHEMBL1979773 | — | Ki | = | 0.7943 | nM | 9.10 |
| CHEMBL1986851 | — | Ki | = | 1.259 | nM | 8.90 |
| CHEMBL1970317 | — | Ki | = | 1.585 | nM | 8.80 |
| CHEMBL379975 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1966514 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1981725 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1981133 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1964692 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1994669 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL1090360 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL371206 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1965988 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL508928 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1979883 | — | Ki | = | 6.31 | nM | 8.20 |
| CHEMBL1973211 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1967531 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL1994321 | — | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL49120 | PD-0166285 | Ki | = | 7.943 | nM | 8.10 |
| CHEMBL2005828 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL1967878 | CENISERTIB | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL2006715 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL2006778 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1991429 | — | Ki | = | 12.59 | nM | 7.90 |
| CHEMBL1981047 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1990885 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1982465 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL5416410 | DASATINIB | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1969190 | — | Ki | = | 15.85 | nM | 7.80 |
| CHEMBL1974328 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1979093 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1979577 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1999484 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL215152 | DEFOSBARASERTIB | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1983111 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1998585 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1966628 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1964948 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1984548 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1984586 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL522892 | DOVITINIB | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL2005509 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL411903 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1992220 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL202721 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1978267 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL271381 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL1999931 | — | Ki | = | 31.62 | nM | 7.50 |