Assay Detail
Functional
CHEMBL1964024
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response validation of uHTS inhibitor hits from DNMT1 for spectral interference using a Fluorescent Molecular Beacon assay. (Class of assay: confirmatory)
200
Total Activities
200
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 200 | 4.30 | 4.69 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1380580 | — | — | 1 | 4.69 |
| CHEMBL1558192 | — | — | 1 | 4.46 |
| CHEMBL1303651 | — | — | 1 | 4.32 |
| CHEMBL1505688 | — | — | 1 | 4.22 |
| CHEMBL224857 | — | — | 1 | 4.09 |
| CHEMBL1472200 | — | — | 1 | 4.03 |
| CHEMBL1361703 | — | — | 1 | - |
| CHEMBL1967046 | — | — | 1 | - |
| CHEMBL583555 | — | — | 1 | - |
| CHEMBL1412087 | — | — | 1 | - |
| CHEMBL1389315 | — | — | 1 | - |
| CHEMBL1414679 | — | — | 1 | - |
| CHEMBL1430983 | — | — | 1 | - |
| CHEMBL1509648 | — | — | 1 | - |
| CHEMBL1523953 | — | — | 1 | - |
| CHEMBL1988862 | — | — | 1 | - |
| CHEMBL1372387 | — | — | 1 | - |
| CHEMBL1967028 | — | — | 1 | - |
| CHEMBL1315592 | — | — | 1 | - |
| CHEMBL1446430 | — | — | 1 | - |
| CHEMBL1358848 | — | — | 1 | - |
| CHEMBL1377441 | — | — | 1 | - |
| CHEMBL1863716 | — | — | 1 | - |
| CHEMBL617 | CEPHALOTHIN | 4.0 | 1 | - |
| CHEMBL1320181 | — | — | 1 | - |
| CHEMBL1536256 | — | — | 1 | - |
| CHEMBL1533351 | — | — | 1 | - |
| CHEMBL1302528 | — | — | 1 | - |
| CHEMBL1423709 | — | — | 1 | - |
| CHEMBL1964442 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1380580 | — | IC50 | = | 20400.0 | nM | 4.69 |
| CHEMBL1558192 | — | IC50 | = | 34400.0 | nM | 4.46 |
| CHEMBL1303651 | — | IC50 | = | 47400.0 | nM | 4.32 |
| CHEMBL1505688 | — | IC50 | = | 60100.0 | nM | 4.22 |
| CHEMBL224857 | — | IC50 | = | 81100.0 | nM | 4.09 |
| CHEMBL1472200 | — | IC50 | = | 93200.0 | nM | 4.03 |
| CHEMBL1510676 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1434555 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1320799 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1440928 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1482590 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1706577 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1730022 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL599013 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1386849 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1975801 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1503050 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1490134 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL233896 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1976649 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1423186 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1612983 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1501577 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1978925 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1511981 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1566530 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1715550 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL494668 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1348946 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL602400 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1603637 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1981657 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1706407 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1397359 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1347385 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1605668 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1480378 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1485277 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1981446 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1408320 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1421559 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1416694 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1453126 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1441143 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1397916 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1469245 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1529522 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1508582 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1514259 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1609276 | — | IC50 | > | 99000.0 | nM | - |