Assay Detail
Functional
CHEMBL1964050
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R): TRFRET-based cell-based high throughput dose response assay to identify nonselective inhibitors of cAMP signaling. (Class of assay: confirmatory)
222
Total Activities
222
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 222 | 4.51 | 4.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1501376 | — | — | 1 | 4.87 |
| CHEMBL1595336 | — | — | 1 | 4.83 |
| CHEMBL1427185 | — | — | 1 | 4.82 |
| CHEMBL1442788 | — | — | 1 | 4.71 |
| CHEMBL1728670 | — | — | 1 | 4.65 |
| CHEMBL1589425 | — | — | 1 | 4.65 |
| CHEMBL1731117 | — | — | 1 | 4.60 |
| CHEMBL1548086 | — | — | 1 | 4.59 |
| CHEMBL1351081 | — | — | 1 | 4.54 |
| CHEMBL790 | CHLORHEXIDINE | 4.0 | 1 | 4.50 |
| CHEMBL1409116 | — | — | 1 | 4.49 |
| CHEMBL1391094 | — | — | 1 | 4.41 |
| CHEMBL1705379 | — | — | 1 | 4.35 |
| CHEMBL1397515 | — | — | 1 | 4.33 |
| CHEMBL2002430 | — | — | 1 | 4.26 |
| CHEMBL1717770 | — | — | 1 | 4.22 |
| CHEMBL1330113 | — | — | 1 | 4.21 |
| CHEMBL1532794 | — | — | 1 | 4.20 |
| CHEMBL1373145 | — | — | 1 | - |
| CHEMBL1548455 | — | — | 1 | - |
| CHEMBL1863528 | — | — | 1 | - |
| CHEMBL1485617 | — | — | 1 | - |
| CHEMBL1985344 | — | — | 1 | - |
| CHEMBL1469994 | — | — | 1 | - |
| CHEMBL1459350 | — | — | 1 | - |
| CHEMBL1494120 | — | — | 1 | - |
| CHEMBL1363895 | — | — | 1 | - |
| CHEMBL1494017 | — | — | 1 | - |
| CHEMBL1491086 | — | — | 1 | - |
| CHEMBL1306085 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1501376 | — | IC50 | = | 13427.0 | nM | 4.87 |
| CHEMBL1595336 | — | IC50 | = | 14860.0 | nM | 4.83 |
| CHEMBL1427185 | — | IC50 | = | 15122.0 | nM | 4.82 |
| CHEMBL1442788 | — | IC50 | = | 19617.0 | nM | 4.71 |
| CHEMBL1728670 | — | IC50 | = | 22600.0 | nM | 4.65 |
| CHEMBL1589425 | — | IC50 | = | 22598.0 | nM | 4.65 |
| CHEMBL1731117 | — | IC50 | = | 25059.0 | nM | 4.60 |
| CHEMBL1548086 | — | IC50 | = | 25909.0 | nM | 4.59 |
| CHEMBL1351081 | — | IC50 | = | 28649.0 | nM | 4.54 |
| CHEMBL790 | CHLORHEXIDINE | IC50 | = | 31818.0 | nM | 4.50 |
| CHEMBL1409116 | — | IC50 | = | 32547.0 | nM | 4.49 |
| CHEMBL1391094 | — | IC50 | = | 39020.0 | nM | 4.41 |
| CHEMBL1705379 | — | IC50 | = | 44672.0 | nM | 4.35 |
| CHEMBL1397515 | — | IC50 | = | 47351.0 | nM | 4.33 |
| CHEMBL2002430 | — | IC50 | = | 55022.0 | nM | 4.26 |
| CHEMBL1717770 | — | IC50 | = | 59809.0 | nM | 4.22 |
| CHEMBL1330113 | — | IC50 | = | 61241.0 | nM | 4.21 |
| CHEMBL1532794 | — | IC50 | = | 63671.0 | nM | 4.20 |
| CHEMBL1458479 | — | IC50 | > | 64561.0 | nM | - |
| CHEMBL1866397 | — | IC50 | > | 64670.0 | nM | - |
| CHEMBL1533937 | — | IC50 | > | 64581.0 | nM | - |
| CHEMBL1300063 | — | IC50 | > | 64571.0 | nM | - |
| CHEMBL1409818 | — | IC50 | > | 64568.0 | nM | - |
| CHEMBL1363112 | — | IC50 | > | 64591.0 | nM | - |
| CHEMBL1997928 | — | IC50 | > | 64573.0 | nM | - |
| CHEMBL153072 | — | IC50 | > | 64555.0 | nM | - |
| CHEMBL1443364 | — | IC50 | > | 64575.0 | nM | - |
| CHEMBL1537104 | — | IC50 | > | 64587.0 | nM | - |
| CHEMBL1372112 | — | IC50 | > | 64551.0 | nM | - |
| CHEMBL1440902 | — | IC50 | > | 64565.0 | nM | - |
| CHEMBL1709842 | — | IC50 | > | 64566.0 | nM | - |
| CHEMBL1310276 | — | IC50 | > | 64591.0 | nM | - |
| CHEMBL1407961 | — | IC50 | > | 64581.0 | nM | - |
| CHEMBL1998496 | — | IC50 | > | 64600.0 | nM | - |
| CHEMBL1514238 | — | IC50 | > | 64595.0 | nM | - |
| CHEMBL1338304 | — | IC50 | > | 64581.0 | nM | - |
| CHEMBL1378309 | — | IC50 | > | 64573.0 | nM | - |
| CHEMBL1715357 | — | IC50 | > | 64585.0 | nM | - |
| CHEMBL1566569 | — | IC50 | > | 64587.0 | nM | - |
| CHEMBL1469171 | — | IC50 | > | 64626.0 | nM | - |
| CHEMBL1725591 | — | IC50 | > | 64566.0 | nM | - |
| CHEMBL1725374 | — | IC50 | > | 64581.0 | nM | - |
| CHEMBL1611832 | — | IC50 | > | 64579.0 | nM | - |
| CHEMBL1422720 | — | IC50 | > | 64546.0 | nM | - |
| CHEMBL1584382 | — | IC50 | > | 64551.0 | nM | - |
| CHEMBL1313430 | — | IC50 | > | 64541.0 | nM | - |
| CHEMBL1979671 | — | IC50 | > | 64562.0 | nM | - |
| CHEMBL1547736 | — | IC50 | > | 64565.0 | nM | - |
| CHEMBL1335878 | — | IC50 | > | 64562.0 | nM | - |
| CHEMBL1977109 | — | IC50 | > | 64622.0 | nM | - |