Assay Detail
Functional
CHEMBL1964113
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Navigating the Kinome. (Class of assay: other) Panel member name: NLK
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | other |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 24 | 7.31 | 8.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1964692 | — | — | 1 | 8.60 |
| CHEMBL272453 | — | — | 1 | 8.40 |
| CHEMBL1968406 | — | — | 1 | 8.30 |
| CHEMBL2000335 | — | — | 1 | 8.30 |
| CHEMBL213505 | — | — | 1 | 7.70 |
| CHEMBL1242373 | — | — | 1 | 7.70 |
| CHEMBL1976220 | — | — | 1 | 7.60 |
| CHEMBL1979093 | — | — | 1 | 7.50 |
| CHEMBL394790 | — | — | 1 | 7.40 |
| CHEMBL1984363 | — | — | 1 | 7.30 |
| CHEMBL262433 | — | — | 1 | 7.20 |
| CHEMBL1994693 | — | — | 1 | 6.90 |
| CHEMBL231209 | — | — | 1 | 6.60 |
| CHEMBL1969190 | — | — | 1 | 6.40 |
| CHEMBL1997349 | — | — | 1 | 6.30 |
| CHEMBL1982135 | — | — | 1 | 6.00 |
| CHEMBL2004365 | — | — | 1 | 6.00 |
| CHEMBL183844 | — | — | 1 | - |
| CHEMBL1970189 | — | — | 1 | - |
| CHEMBL1965570 | — | — | 1 | - |
| CHEMBL1980163 | — | — | 1 | - |
| CHEMBL1971649 | — | — | 1 | - |
| CHEMBL1972489 | — | — | 1 | - |
| CHEMBL1990912 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1964692 | — | Ki | = | 2.512 | nM | 8.60 |
| CHEMBL272453 | — | Ki | = | 3.981 | nM | 8.40 |
| CHEMBL1968406 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL2000335 | — | Ki | = | 5.012 | nM | 8.30 |
| CHEMBL213505 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1242373 | — | Ki | = | 19.95 | nM | 7.70 |
| CHEMBL1976220 | — | Ki | = | 25.12 | nM | 7.60 |
| CHEMBL1979093 | — | Ki | = | 31.62 | nM | 7.50 |
| CHEMBL394790 | — | Ki | = | 39.81 | nM | 7.40 |
| CHEMBL1984363 | — | Ki | = | 50.12 | nM | 7.30 |
| CHEMBL262433 | — | Ki | = | 63.1 | nM | 7.20 |
| CHEMBL1994693 | — | Ki | = | 125.89 | nM | 6.90 |
| CHEMBL231209 | — | Ki | = | 251.19 | nM | 6.60 |
| CHEMBL1969190 | — | Ki | = | 398.11 | nM | 6.40 |
| CHEMBL1997349 | — | Ki | = | 501.19 | nM | 6.30 |
| CHEMBL1982135 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL2004365 | — | Ki | = | 1000.0 | nM | 6.00 |
| CHEMBL183844 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1970189 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1965570 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1980163 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1971649 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1972489 | — | Ki | > | 1584.89 | nM | - |
| CHEMBL1990912 | — | Ki | > | 1584.89 | nM | - |