Assay Detail
Binding
CHEMBL2162865
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Inhibition of USP47 by Ub-CHOP reporter assay
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Ubiquitin carboxyl-terminal hydrolase 47 (CHEMBL2157851) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Selective Dual Inhibitors of the Cancer-Related Deubiquitylating Proteases USP7 and USP47.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 5.73 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2159507 | — | — | 1 | 6.46 |
| CHEMBL2159505 | — | — | 1 | 6.30 |
| CHEMBL2159503 | — | — | 1 | 6.28 |
| CHEMBL2159504 | — | — | 1 | 6.06 |
| CHEMBL2159508 | — | — | 1 | 6.00 |
| CHEMBL2159500 | — | — | 1 | 5.92 |
| CHEMBL2159501 | — | — | 1 | 5.89 |
| CHEMBL2159499 | — | — | 1 | 5.66 |
| CHEMBL2159497 | — | — | 1 | 5.43 |
| CHEMBL2159495 | — | — | 1 | 5.37 |
| CHEMBL2159502 | — | — | 1 | 5.26 |
| CHEMBL2159498 | — | — | 1 | 5.06 |
| CHEMBL2159496 | — | — | 1 | 4.85 |
| CHEMBL2159506 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2159507 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL2159505 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL2159503 | — | IC50 | = | 530.0 | nM | 6.28 |
| CHEMBL2159504 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL2159508 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL2159500 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL2159501 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL2159499 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL2159497 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL2159495 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL2159502 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL2159498 | — | IC50 | = | 8700.0 | nM | 5.06 |
| CHEMBL2159496 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL2159506 | — | IC50 | > | 31600.0 | nM | - |