Assay Detail
Binding
CHEMBL2184660
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human SRB1-mediated Hepatitis C virus genotype 2a entry into human HuH7.5 cells by luciferase reporter gene assay
35
Total Activities
34
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Huh-7 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Scavenger receptor class B member 1 (CHEMBL1914272) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of ITX 4520: a highly potent orally bioavailable hepatitis C virus entry inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 8.16 | 8.82 |
| IC90 | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1914885 | — | — | 1 | 8.82 |
| CHEMBL2179502 | — | — | 1 | 8.82 |
| CHEMBL2179514 | — | — | 1 | 8.82 |
| CHEMBL2179515 | — | — | 1 | 8.82 |
| CHEMBL2179485 | — | — | 1 | 8.82 |
| CHEMBL2179509 | — | — | 1 | 8.82 |
| CHEMBL2179511 | — | — | 1 | 8.82 |
| CHEMBL2179508 | — | — | 1 | 8.82 |
| CHEMBL2179507 | — | — | 1 | 8.82 |
| CHEMBL2179504 | — | — | 1 | 8.82 |
| CHEMBL2179510 | — | — | 2 | 8.82 |
| CHEMBL2179501 | — | — | 1 | 8.82 |
| CHEMBL2179500 | — | — | 1 | 8.82 |
| CHEMBL2179499 | — | — | 1 | 8.82 |
| CHEMBL2179493 | — | — | 1 | 8.82 |
| CHEMBL2179497 | — | — | 1 | 8.30 |
| CHEMBL2179512 | — | — | 1 | 8.30 |
| CHEMBL2179106 | — | — | 1 | 8.30 |
| CHEMBL2179488 | — | — | 1 | 8.00 |
| CHEMBL2177128 | — | — | 1 | 7.82 |
| CHEMBL2179487 | — | — | 1 | 7.82 |
| CHEMBL2179486 | — | — | 1 | 7.82 |
| CHEMBL2179494 | — | — | 1 | 7.82 |
| CHEMBL2179498 | — | — | 1 | 7.82 |
| CHEMBL2179506 | — | — | 1 | 7.82 |
| CHEMBL2179513 | — | — | 1 | 7.82 |
| CHEMBL2179490 | — | — | 1 | 7.52 |
| CHEMBL2179496 | — | — | 1 | 7.30 |
| CHEMBL2179495 | — | — | 1 | 7.30 |
| CHEMBL2179503 | — | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2179499 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179500 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179501 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179502 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179504 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179507 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179508 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179510 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179511 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179493 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179514 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179515 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179485 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL1914885 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179509 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL2179106 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL2179512 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL2179497 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL2179488 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL2179486 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179513 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179506 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179498 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2177128 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179494 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179487 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL2179490 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL2179503 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179496 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179495 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179505 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179492 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179489 | — | IC50 | = | 50.0 | nM | 7.30 |
| CHEMBL2179491 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL2179510 | — | IC90 | = | 50.0 | nM | - |