Assay Detail
Functional
CHEMBL2214244
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Cytotoxicity against human HL60 cells after 48 hrs by MTT assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Cytotoxic alkaloids from the whole plants of Zephyranthes candida.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.95 | 6.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2208199 | — | — | 1 | 6.09 |
| CHEMBL2208203 | — | — | 1 | 6.04 |
| CHEMBL401114 | (+)-HAEMANTHAMINE | — | 1 | 5.85 |
| CHEMBL400092 | LYCORINE | — | 1 | 5.80 |
| CHEMBL2208202 | NIGRAGILLIN | — | 1 | - |
| CHEMBL2005884 | — | — | 1 | - |
| CHEMBL511443 | TRISPHAERIDINE | — | 1 | - |
| CHEMBL2208201 | — | — | 1 | - |
| CHEMBL2208200 | — | — | 1 | - |
| CHEMBL2208198 | — | — | 1 | - |
| CHEMBL2208206 | — | — | 1 | - |
| CHEMBL2208205 | — | — | 1 | - |
| CHEMBL2208204 | — | — | 1 | - |
| CHEMBL457605 | TAZETTINE | — | 1 | - |
| CHEMBL1976572 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2208199 | — | IC50 | = | 810.0 | nM | 6.09 |
| CHEMBL2208203 | — | IC50 | = | 910.0 | nM | 6.04 |
| CHEMBL401114 | (+)-HAEMANTHAMINE | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL400092 | LYCORINE | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL2208202 | NIGRAGILLIN | IC50 | > | 10000.0 | nM | - |
| CHEMBL2005884 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL511443 | TRISPHAERIDINE | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208201 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208200 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208198 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208206 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208205 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL2208204 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL457605 | TAZETTINE | IC50 | > | 10000.0 | nM | - |
| CHEMBL1976572 | — | IC50 | > | 10000.0 | nM | - |