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Assay Detail

CHEMBL2328232

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Junin virus pseudovirions infected in HEK293T/17 cells after 72 hrs by luciferase reporter gene assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mammarenavirus juninense
Cell Type HEK-293T
Confidence 1 — Organism
Curated By Autocuration

Target

Junin virus (CHEMBL4523072)
Type ORGANISM
Organism Mammarenavirus juninense

Publication

Discovery and optimization of potent broad-spectrum arenavirus inhibitors derived from benzimidazole.
Dai D, Burgeson JR, Gharaibeh DN, Moore AL, Larson RA, Cerruti NR, Amberg SM, Bolken TC, Hruby DE.
Bioorg Med Chem Lett (2013) 23 : 744 -749
PubMed 23265895 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 8.36 9.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2314859 1 9.21
CHEMBL2322820 1 8.30
CHEMBL2322826 1 8.11
CHEMBL2322822 1 7.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2314859 EC50 = 0.62 nM 9.21
CHEMBL2322820 EC50 = 5.0 nM 8.30
CHEMBL2322826 EC50 = 7.7 nM 8.11
CHEMBL2322822 EC50 = 16.0 nM 7.80