Assay Detail
Functional
CHEMBL2363152
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SANGER: Inhibition of human CTB-1 cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CTB-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.65 | 9.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.37 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.79 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.72 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.53 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.08 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.06 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.01 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.79 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.77 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.70 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.61 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 7.57 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.46 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.27 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.19 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.12 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.11 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.88 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.87 |
| CHEMBL300389 | — | — | 1 | 6.82 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.76 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.65 |
| CHEMBL379975 | — | — | 1 | 6.62 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.61 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.57 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.51 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.49 |
| CHEMBL514499 | GW843682X | — | 1 | 6.44 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.39 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.37 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.4292 | nM | 9.37 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.636 | nM | 8.79 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.922 | nM | 8.72 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 2.934 | nM | 8.53 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 8.305 | nM | 8.08 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 8.64 | nM | 8.06 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 9.673 | nM | 8.01 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 16.23 | nM | 7.79 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 16.97 | nM | 7.77 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 19.8 | nM | 7.70 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 24.67 | nM | 7.61 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 26.94 | nM | 7.57 |
| CHEMBL803 | CYTARABINE | IC50 | = | 34.4 | nM | 7.46 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 53.39 | nM | 7.27 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 64.19 | nM | 7.19 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 75.88 | nM | 7.12 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 78.1 | nM | 7.11 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 133.25 | nM | 6.88 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 134.69 | nM | 6.87 |
| CHEMBL300389 | — | IC50 | = | 152.6 | nM | 6.82 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 173.16 | nM | 6.76 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 222.28 | nM | 6.65 |
| CHEMBL379975 | — | IC50 | = | 242.09 | nM | 6.62 |
| CHEMBL513909 | BI-2536 | IC50 | = | 244.93 | nM | 6.61 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 272.15 | nM | 6.57 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 306.37 | nM | 6.51 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 327.53 | nM | 6.49 |
| CHEMBL514499 | GW843682X | IC50 | = | 360.72 | nM | 6.44 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 405.02 | nM | 6.39 |
| CHEMBL939 | GEFITINIB | IC50 | = | 424.4 | nM | 6.37 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 497.45 | nM | 6.30 |
| CHEMBL379300 | A-443654 | IC50 | = | 508.66 | nM | 6.29 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 537.92 | nM | 6.27 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 548.2 | nM | 6.26 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 605.98 | nM | 6.22 |
| CHEMBL64925 | MG-132 | IC50 | = | 779.55 | nM | 6.11 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 859.02 | nM | 6.07 |
| CHEMBL585951 | — | IC50 | = | 1106.32 | nM | 5.96 |
| CHEMBL188678 | — | IC50 | = | 1115.46 | nM | 5.95 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 1142.93 | nM | 5.94 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 1289.9 | nM | 5.89 |
| CHEMBL591429 | PAC-1 | IC50 | = | 1436.87 | nM | 5.84 |
| CHEMBL573107 | — | IC50 | = | 1446.79 | nM | 5.84 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1486.0 | nM | 5.83 |
| CHEMBL515416 | — | IC50 | = | 1620.19 | nM | 5.79 |
| CHEMBL38 | TRETINOIN | IC50 | = | 1603.89 | nM | 5.79 |
| CHEMBL202721 | — | IC50 | = | 1670.82 | nM | 5.78 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1687.66 | nM | 5.77 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 2022.46 | nM | 5.69 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 2296.43 | nM | 5.64 |