Assay Detail
Functional
CHEMBL2363223
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SANGER: Inhibition of human EW-13 cell growth in a cell viability assay.
130
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | EW-13 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 130 | 5.58 | 10.95 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 10.95 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.04 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.64 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.49 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.29 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.18 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 8.02 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.84 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.70 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.65 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.54 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.44 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.36 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.28 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.14 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 7.11 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 7.05 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.02 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.65 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.57 |
| CHEMBL585951 | — | — | 1 | 6.53 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.53 |
| CHEMBL259181 | — | — | 1 | 6.38 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.36 |
| CHEMBL1023 | BEXAROTENE | 4.0 | 1 | 6.31 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 6.23 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.17 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.04 |
| CHEMBL300389 | — | — | 1 | 5.89 |
| CHEMBL1190711 | — | — | 1 | 5.83 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.01122 | nM | 10.95 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.9028 | nM | 9.04 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 2.309 | nM | 8.64 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 3.267 | nM | 8.49 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 5.179 | nM | 8.29 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 6.617 | nM | 8.18 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 9.626 | nM | 8.02 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 14.54 | nM | 7.84 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 19.75 | nM | 7.70 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 22.53 | nM | 7.65 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 29.04 | nM | 7.54 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 36.52 | nM | 7.44 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 44.06 | nM | 7.36 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 52.51 | nM | 7.28 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 72.3 | nM | 7.14 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 77.76 | nM | 7.11 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 88.85 | nM | 7.05 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 95.75 | nM | 7.02 |
| CHEMBL939 | GEFITINIB | IC50 | = | 225.1 | nM | 6.65 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 266.74 | nM | 6.57 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 292.08 | nM | 6.53 |
| CHEMBL585951 | — | IC50 | = | 297.05 | nM | 6.53 |
| CHEMBL259181 | — | IC50 | = | 412.84 | nM | 6.38 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 435.48 | nM | 6.36 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 485.1 | nM | 6.31 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 583.41 | nM | 6.23 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 667.79 | nM | 6.17 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 909.0 | nM | 6.04 |
| CHEMBL300389 | — | IC50 | = | 1274.77 | nM | 5.89 |
| CHEMBL1190711 | — | IC50 | = | 1473.33 | nM | 5.83 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 1634.66 | nM | 5.79 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1981.5 | nM | 5.70 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 2468.35 | nM | 5.61 |
| CHEMBL105442 | CI-1040 | IC50 | = | 2563.39 | nM | 5.59 |
| CHEMBL379300 | A-443654 | IC50 | = | 2666.58 | nM | 5.57 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 2687.68 | nM | 5.57 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 3015.58 | nM | 5.52 |
| CHEMBL514499 | GW843682X | IC50 | = | 3053.61 | nM | 5.51 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3525.1 | nM | 5.45 |
| CHEMBL513909 | BI-2536 | IC50 | = | 3834.17 | nM | 5.42 |
| CHEMBL472940 | — | IC50 | = | 4201.48 | nM | 5.38 |
| CHEMBL379975 | — | IC50 | = | 4198.83 | nM | 5.38 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 4166.46 | nM | 5.38 |
| CHEMBL472004 | — | IC50 | = | 5168.72 | nM | 5.29 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 5766.27 | nM | 5.24 |
| CHEMBL2363137 | — | IC50 | = | 6038.5 | nM | 5.22 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 6476.92 | nM | 5.19 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 6774.24 | nM | 5.17 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 7351.62 | nM | 5.13 |
| CHEMBL38 | TRETINOIN | IC50 | = | 7610.78 | nM | 5.12 |