Assay Detail
Functional
CHEMBL2363251
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SANGER: Inhibition of human H9 cell growth in a cell viability assay.
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | H9 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 40 | 6.45 | 9.45 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.45 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.90 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.65 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 8.31 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 8.24 |
| CHEMBL3349342 | — | — | 1 | 7.70 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 7.64 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 7.64 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.46 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.36 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.24 |
| CHEMBL573107 | — | — | 1 | 7.22 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 7.17 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 7.15 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.92 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.86 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.59 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.41 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.41 |
| CHEMBL477989 | SB590885 | — | 1 | 6.40 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 6.36 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.30 |
| CHEMBL379975 | — | — | 1 | 6.08 |
| CHEMBL202721 | — | — | 1 | 6.03 |
| CHEMBL189584 | PD-173074 | — | 1 | 5.67 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 5.56 |
| CHEMBL11359 | CISPLATIN | 4.0 | 1 | 5.44 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.43 |
| CHEMBL572881 | MOTESANIB | 3.0 | 1 | 5.09 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 4.90 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.3582 | nM | 9.45 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.245 | nM | 8.90 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 2.248 | nM | 8.65 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 4.88 | nM | 8.31 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 5.768 | nM | 8.24 |
| CHEMBL3349342 | — | IC50 | = | 20.08 | nM | 7.70 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 22.88 | nM | 7.64 |
| CHEMBL105442 | CI-1040 | IC50 | = | 22.76 | nM | 7.64 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 34.78 | nM | 7.46 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 43.71 | nM | 7.36 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 58.13 | nM | 7.24 |
| CHEMBL573107 | — | IC50 | = | 60.19 | nM | 7.22 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 66.92 | nM | 7.17 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 71.32 | nM | 7.15 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 121.65 | nM | 6.92 |
| CHEMBL939 | GEFITINIB | IC50 | = | 137.2 | nM | 6.86 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 255.04 | nM | 6.59 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 388.83 | nM | 6.41 |
| CHEMBL803 | CYTARABINE | IC50 | = | 391.42 | nM | 6.41 |
| CHEMBL477989 | SB590885 | IC50 | = | 401.02 | nM | 6.40 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 434.64 | nM | 6.36 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 495.43 | nM | 6.30 |
| CHEMBL379975 | — | IC50 | = | 831.5 | nM | 6.08 |
| CHEMBL202721 | — | IC50 | = | 929.79 | nM | 6.03 |
| CHEMBL189584 | PD-173074 | IC50 | = | 2143.06 | nM | 5.67 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 2737.93 | nM | 5.56 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 3647.42 | nM | 5.44 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 3671.44 | nM | 5.43 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 8127.32 | nM | 5.09 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 12557.75 | nM | 4.90 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 13847.53 | nM | 4.86 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 16626.02 | nM | 4.78 |
| CHEMBL506871 | VELIPARIB | IC50 | = | 18283.32 | nM | 4.74 |
| CHEMBL240954 | — | IC50 | = | 22289.26 | nM | 4.65 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 31300.81 | nM | 4.50 |
| CHEMBL393929 | — | IC50 | = | 51092.97 | nM | 4.29 |
| CHEMBL210618 | — | IC50 | = | 84492.01 | nM | 4.07 |
| CHEMBL103667 | DORAMAPIMOD | IC50 | = | 177641.06 | nM | - |
| CHEMBL176544 | — | IC50 | = | 135377.48 | nM | - |
| CHEMBL1431 | METFORMIN | IC50 | = | 7136123.64 | nM | - |