Assay Detail
Functional
CHEMBL2363460
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SANGER: Inhibition of human NB7 cell growth in a cell viability assay.
101
Total Activities
100
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NB7 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 101 | 5.37 | 7.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.91 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.84 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 7.80 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.78 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.75 |
| CHEMBL217354 | — | — | 1 | 7.53 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 7.08 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 6.87 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.72 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.71 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.46 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.41 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 6.35 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.32 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.26 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 6.09 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.08 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.05 |
| CHEMBL188678 | — | — | 1 | 5.90 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 5.82 |
| CHEMBL202721 | — | — | 1 | 5.76 |
| CHEMBL300389 | — | — | 1 | 5.75 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.70 |
| CHEMBL509032 | TAE-684 | — | 1 | 5.70 |
| CHEMBL176544 | — | — | 1 | 5.70 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 5.66 |
| CHEMBL210618 | — | — | 1 | 5.64 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.64 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 5.63 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 12.43 | nM | 7.91 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 14.39 | nM | 7.84 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 15.92 | nM | 7.80 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 16.8 | nM | 7.78 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 17.88 | nM | 7.75 |
| CHEMBL217354 | — | IC50 | = | 29.28 | nM | 7.53 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 82.31 | nM | 7.08 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 134.39 | nM | 6.87 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 189.89 | nM | 6.72 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 195.12 | nM | 6.71 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 345.74 | nM | 6.46 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 389.83 | nM | 6.41 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 447.6 | nM | 6.35 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 477.46 | nM | 6.32 |
| CHEMBL939 | GEFITINIB | IC50 | = | 546.32 | nM | 6.26 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 814.14 | nM | 6.09 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 824.11 | nM | 6.08 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 899.42 | nM | 6.05 |
| CHEMBL188678 | — | IC50 | = | 1247.45 | nM | 5.90 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1515.52 | nM | 5.82 |
| CHEMBL202721 | — | IC50 | = | 1752.97 | nM | 5.76 |
| CHEMBL300389 | — | IC50 | = | 1765.25 | nM | 5.75 |
| CHEMBL509032 | TAE-684 | IC50 | = | 2005.55 | nM | 5.70 |
| CHEMBL176544 | — | IC50 | = | 1981.37 | nM | 5.70 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1993.23 | nM | 5.70 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 2196.73 | nM | 5.66 |
| CHEMBL210618 | — | IC50 | = | 2274.73 | nM | 5.64 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 2296.76 | nM | 5.64 |
| CHEMBL105442 | CI-1040 | IC50 | = | 2340.86 | nM | 5.63 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 2921.39 | nM | 5.53 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 4403.76 | nM | 5.36 |
| CHEMBL3349342 | — | IC50 | = | 4705.34 | nM | 5.33 |
| CHEMBL64925 | MG-132 | IC50 | = | 5045.89 | nM | 5.30 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 5141.12 | nM | 5.29 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 6213.73 | nM | 5.21 |
| CHEMBL379300 | A-443654 | IC50 | = | 6641.85 | nM | 5.18 |
| CHEMBL1186585 | — | IC50 | = | 8636.53 | nM | 5.06 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 10752.58 | nM | 4.97 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 11329.69 | nM | 4.95 |
| CHEMBL477989 | SB590885 | IC50 | = | 11895.59 | nM | 4.92 |
| CHEMBL515416 | — | IC50 | = | 12483.85 | nM | 4.90 |
| CHEMBL554 | LAPATINIB | IC50 | = | 14237.45 | nM | 4.85 |
| CHEMBL577784 | BX-795 | IC50 | = | 13981.23 | nM | 4.85 |
| CHEMBL1242367 | — | IC50 | = | 14504.52 | nM | 4.84 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 14965.24 | nM | 4.83 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 15361.0 | nM | 4.81 |
| CHEMBL473417 | VISMODEGIB | IC50 | = | 15891.02 | nM | 4.80 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 16697.05 | nM | 4.78 |
| CHEMBL513909 | BI-2536 | IC50 | = | 17746.71 | nM | 4.75 |
| CHEMBL573107 | — | IC50 | = | 19175.3 | nM | 4.72 |