Assay Detail
Functional
CHEMBL2363496
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SANGER: Inhibition of human NCI-H1975 cell growth in a cell viability assay.
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H1975 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.05 | 7.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.62 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.48 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.21 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.90 |
| CHEMBL217354 | — | — | 1 | 5.86 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 5.77 |
| CHEMBL399530 | — | — | 1 | 5.55 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 5.19 |
| CHEMBL2137530 | SERDEMETAN | 2.0 | 1 | 4.71 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 4.67 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 4.62 |
| CHEMBL1090771 | AVAGACESTAT | 2.0 | 1 | 4.56 |
| CHEMBL176544 | — | — | 1 | 4.55 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 1 | 4.52 |
| CHEMBL102714 | SB-216763 | — | 1 | 4.49 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 4.45 |
| CHEMBL1186585 | — | — | 1 | 4.39 |
| CHEMBL2134202 | — | — | 1 | 4.27 |
| CHEMBL1173055 | RUCAPARIB | 4.0 | 1 | 4.24 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 4.04 |
| CHEMBL1090090 | VX-702 | 2.0 | 1 | 4.01 |
| CHEMBL473417 | VISMODEGIB | 4.0 | 1 | - |
| CHEMBL255342 | — | — | 1 | - |
| CHEMBL848 | LENALIDOMIDE | 4.0 | 1 | - |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | - |
| CHEMBL38 | TRETINOIN | 4.0 | 1 | - |
| CHEMBL11359 | CISPLATIN | 4.0 | 1 | - |
| CHEMBL483849 | — | — | 1 | - |
| CHEMBL1431 | METFORMIN | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL159 | VINBLASTINE | IC50 | = | 24.23 | nM | 7.62 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 334.48 | nM | 6.48 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 617.28 | nM | 6.21 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1250.41 | nM | 5.90 |
| CHEMBL217354 | — | IC50 | = | 1375.86 | nM | 5.86 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 1696.85 | nM | 5.77 |
| CHEMBL399530 | — | IC50 | = | 2815.37 | nM | 5.55 |
| CHEMBL105442 | CI-1040 | IC50 | = | 6472.15 | nM | 5.19 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 19551.17 | nM | 4.71 |
| CHEMBL939 | GEFITINIB | IC50 | = | 21461.01 | nM | 4.67 |
| CHEMBL803 | CYTARABINE | IC50 | = | 23880.66 | nM | 4.62 |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 27450.05 | nM | 4.56 |
| CHEMBL176544 | — | IC50 | = | 28165.2 | nM | 4.55 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 29911.62 | nM | 4.52 |
| CHEMBL102714 | SB-216763 | IC50 | = | 32358.25 | nM | 4.49 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 35902.04 | nM | 4.45 |
| CHEMBL1186585 | — | IC50 | = | 40952.34 | nM | 4.39 |
| CHEMBL2134202 | — | IC50 | = | 53896.63 | nM | 4.27 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 58264.62 | nM | 4.24 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 92137.59 | nM | 4.04 |
| CHEMBL1090090 | VX-702 | IC50 | = | 96550.29 | nM | 4.01 |
| CHEMBL473417 | VISMODEGIB | IC50 | = | 568681.77 | nM | - |
| CHEMBL255342 | — | IC50 | = | 245623.53 | nM | - |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 238657.39 | nM | - |
| CHEMBL255863 | NILOTINIB | IC50 | = | 131950.78 | nM | - |
| CHEMBL38 | TRETINOIN | IC50 | = | 218983.42 | nM | - |
| CHEMBL11359 | CISPLATIN | IC50 | = | 408911.19 | nM | - |
| CHEMBL483849 | — | IC50 | = | 1071537.7 | nM | - |
| CHEMBL1431 | METFORMIN | IC50 | = | 11679261.19 | nM | - |