Assay Detail
Functional
CHEMBL2363554
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human NCI-SNU-16 cell growth in a cell viability assay.
78
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SNU-16 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 78 | 5.48 | 8.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.12 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.00 |
| CHEMBL213100 | — | — | 1 | 7.80 |
| CHEMBL514499 | GW843682X | — | 1 | 7.69 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.51 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.41 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 6.97 |
| CHEMBL300389 | — | — | 1 | 6.87 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.72 |
| CHEMBL1256459 | TORIN1 | — | 1 | 6.52 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 6.20 |
| CHEMBL509032 | TAE-684 | — | 1 | 6.14 |
| CHEMBL401930 | — | — | 1 | 6.06 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 5.84 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 5.83 |
| CHEMBL379300 | A-443654 | — | 1 | 5.76 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 5.25 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.17 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 5.17 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 5.07 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 5.04 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 5.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 4.88 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 4.81 |
| CHEMBL1673039 | — | — | 1 | 4.73 |
| CHEMBL180127 | SALUBRINAL | — | 1 | 4.68 |
| CHEMBL2144069 | — | — | 1 | 4.56 |
| CHEMBL197603 | — | — | 1 | 4.52 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 4.51 |
| CHEMBL64925 | MG-132 | — | 2 | 4.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 7.653 | nM | 8.12 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 10.08 | nM | 8.00 |
| CHEMBL213100 | — | IC50 | = | 15.72 | nM | 7.80 |
| CHEMBL514499 | GW843682X | IC50 | = | 20.47 | nM | 7.69 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 31.0 | nM | 7.51 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 38.56 | nM | 7.41 |
| CHEMBL513909 | BI-2536 | IC50 | = | 107.42 | nM | 6.97 |
| CHEMBL300389 | — | IC50 | = | 135.67 | nM | 6.87 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 189.01 | nM | 6.72 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 302.05 | nM | 6.52 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 635.71 | nM | 6.20 |
| CHEMBL509032 | TAE-684 | IC50 | = | 726.64 | nM | 6.14 |
| CHEMBL401930 | — | IC50 | = | 873.27 | nM | 6.06 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1434.51 | nM | 5.84 |
| CHEMBL535 | SUNITINIB | IC50 | = | 1464.86 | nM | 5.83 |
| CHEMBL379300 | A-443654 | IC50 | = | 1728.12 | nM | 5.76 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 5640.74 | nM | 5.25 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 6746.7 | nM | 5.17 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 6743.09 | nM | 5.17 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 8561.28 | nM | 5.07 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 9210.26 | nM | 5.04 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 9794.95 | nM | 5.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 13125.83 | nM | 4.88 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 15463.28 | nM | 4.81 |
| CHEMBL1673039 | — | IC50 | = | 18800.19 | nM | 4.73 |
| CHEMBL180127 | SALUBRINAL | IC50 | = | 21053.92 | nM | 4.68 |
| CHEMBL2144069 | — | IC50 | = | 27779.52 | nM | 4.56 |
| CHEMBL197603 | — | IC50 | = | 30303.61 | nM | 4.52 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 31183.65 | nM | 4.51 |
| CHEMBL64925 | MG-132 | IC50 | = | 38565.34 | nM | 4.41 |
| CHEMBL64925 | MG-132 | IC50 | = | 40777.11 | nM | 4.39 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 48314.18 | nM | 4.32 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 49214.29 | nM | 4.31 |
| CHEMBL515416 | — | IC50 | = | 50965.86 | nM | 4.29 |
| CHEMBL553 | ERLOTINIB | IC50 | = | 62009.65 | nM | 4.21 |
| CHEMBL1190711 | — | IC50 | = | 61741.48 | nM | 4.21 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 73628.56 | nM | 4.13 |
| CHEMBL1643959 | — | IC50 | = | 82958.05 | nM | 4.08 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 96355.36 | nM | 4.02 |
| CHEMBL4298697 | — | IC50 | = | 97262.74 | nM | 4.01 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 2384689.01 | nM | - |
| CHEMBL2363137 | — | IC50 | = | 208999.53 | nM | - |
| CHEMBL591429 | PAC-1 | IC50 | = | 251304.16 | nM | - |
| CHEMBL472940 | — | IC50 | = | 4266111.35 | nM | - |
| CHEMBL558642 | GSK-650394 | IC50 | = | 3269632.92 | nM | - |
| CHEMBL1242367 | — | IC50 | = | 135180.38 | nM | - |
| CHEMBL483847 | — | IC50 | = | 221460.45 | nM | - |
| CHEMBL217092 | SARACATINIB | IC50 | = | 371335.14 | nM | - |
| CHEMBL575448 | BMS-754807 | IC50 | = | 431867.14 | nM | - |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 752686.65 | nM | - |