Assay Detail
Functional
CHEMBL2363562
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SANGER: Inhibition of human NTERA-S-cl-D1 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NTERA-2-cl-D1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.99 | 10.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 10.66 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 9.86 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.61 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.56 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.38 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 9.35 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.14 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.11 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 9.03 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 8.86 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.79 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.68 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.23 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.87 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 7.84 |
| CHEMBL514499 | GW843682X | — | 1 | 7.76 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.71 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.68 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 7.60 |
| CHEMBL379300 | A-443654 | — | 1 | 7.56 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.49 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.47 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.37 |
| CHEMBL300389 | — | — | 1 | 7.29 |
| CHEMBL64925 | MG-132 | — | 2 | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.98 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.91 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.84 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.80 |
| CHEMBL217354 | — | — | 1 | 6.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL105 | MITOMYCIN | IC50 | = | 0.02213 | nM | 10.66 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 0.1391 | nM | 9.86 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.2434 | nM | 9.61 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.2738 | nM | 9.56 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.4124 | nM | 9.38 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 0.443 | nM | 9.35 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7182 | nM | 9.14 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.7726 | nM | 9.11 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 0.9386 | nM | 9.03 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 1.37 | nM | 8.86 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1.641 | nM | 8.79 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 2.088 | nM | 8.68 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.893 | nM | 8.23 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 13.39 | nM | 7.87 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 14.34 | nM | 7.84 |
| CHEMBL514499 | GW843682X | IC50 | = | 17.36 | nM | 7.76 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 19.39 | nM | 7.71 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 20.69 | nM | 7.68 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 25.02 | nM | 7.60 |
| CHEMBL379300 | A-443654 | IC50 | = | 27.59 | nM | 7.56 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 32.26 | nM | 7.49 |
| CHEMBL513909 | BI-2536 | IC50 | = | 33.99 | nM | 7.47 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 43.0 | nM | 7.37 |
| CHEMBL300389 | — | IC50 | = | 50.84 | nM | 7.29 |
| CHEMBL64925 | MG-132 | IC50 | = | 57.72 | nM | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 104.48 | nM | 6.98 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 122.83 | nM | 6.91 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 143.57 | nM | 6.84 |
| CHEMBL803 | CYTARABINE | IC50 | = | 159.1 | nM | 6.80 |
| CHEMBL217354 | — | IC50 | = | 166.68 | nM | 6.78 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 177.78 | nM | 6.75 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 189.62 | nM | 6.72 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 201.13 | nM | 6.70 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 208.95 | nM | 6.68 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 237.44 | nM | 6.62 |
| CHEMBL401930 | — | IC50 | = | 257.49 | nM | 6.59 |
| CHEMBL213100 | — | IC50 | = | 288.55 | nM | 6.54 |
| CHEMBL585951 | — | IC50 | = | 315.67 | nM | 6.50 |
| CHEMBL509032 | TAE-684 | IC50 | = | 333.96 | nM | 6.48 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 328.36 | nM | 6.48 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 362.97 | nM | 6.44 |
| CHEMBL64925 | MG-132 | IC50 | = | 425.92 | nM | 6.37 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 500.19 | nM | 6.30 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 700.63 | nM | 6.16 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 848.5 | nM | 6.07 |
| CHEMBL577784 | BX-795 | IC50 | = | 1077.75 | nM | 5.97 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 1243.46 | nM | 5.91 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1317.61 | nM | 5.88 |
| CHEMBL521686 | OLAPARIB | IC50 | = | 1333.41 | nM | 5.88 |
| CHEMBL2363137 | — | IC50 | = | 1428.13 | nM | 5.84 |