Assay Detail
Functional
CHEMBL2363585
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SANGER: Inhibition of human PANC-08-13 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PANC-08-13 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.44 | 8.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 8.06 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.02 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.62 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.61 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.51 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.35 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.33 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.24 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.21 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.11 |
| CHEMBL585951 | — | — | 1 | 7.05 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.50 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.27 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.24 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.18 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.16 |
| CHEMBL1091644 | LINSITINIB | 3.0 | 1 | 6.06 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.93 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.87 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.87 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 5.86 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.79 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 5.63 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.62 |
| CHEMBL188678 | — | — | 1 | 5.47 |
| CHEMBL191384 | — | — | 1 | 5.44 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 5.44 |
| CHEMBL217354 | — | — | 1 | 5.42 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.42 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 5.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL575448 | BMS-754807 | IC50 | = | 8.604 | nM | 8.06 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 9.634 | nM | 8.02 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 23.81 | nM | 7.62 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 24.65 | nM | 7.61 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 31.13 | nM | 7.51 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 44.89 | nM | 7.35 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 46.95 | nM | 7.33 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 58.01 | nM | 7.24 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 61.47 | nM | 7.21 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 77.16 | nM | 7.11 |
| CHEMBL585951 | — | IC50 | = | 89.99 | nM | 7.05 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 320.22 | nM | 6.50 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 531.77 | nM | 6.27 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 573.89 | nM | 6.24 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 660.68 | nM | 6.18 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 694.99 | nM | 6.16 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 863.77 | nM | 6.06 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 1164.16 | nM | 5.93 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1345.86 | nM | 5.87 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1338.03 | nM | 5.87 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 1396.13 | nM | 5.86 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 1630.84 | nM | 5.79 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 2332.35 | nM | 5.63 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 2397.77 | nM | 5.62 |
| CHEMBL188678 | — | IC50 | = | 3412.78 | nM | 5.47 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 3634.72 | nM | 5.44 |
| CHEMBL191384 | — | IC50 | = | 3632.22 | nM | 5.44 |
| CHEMBL217354 | — | IC50 | = | 3765.65 | nM | 5.42 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3796.02 | nM | 5.42 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 3886.13 | nM | 5.41 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 4077.3 | nM | 5.39 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 4804.63 | nM | 5.32 |
| CHEMBL176544 | — | IC50 | = | 5873.58 | nM | 5.23 |
| CHEMBL803 | CYTARABINE | IC50 | = | 7781.08 | nM | 5.11 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 10430.49 | nM | 4.98 |
| CHEMBL1190711 | — | IC50 | = | 10542.71 | nM | 4.98 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 12052.11 | nM | 4.92 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 12629.84 | nM | 4.90 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 14910.85 | nM | 4.83 |
| CHEMBL577784 | BX-795 | IC50 | = | 15195.89 | nM | 4.82 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 15685.87 | nM | 4.80 |
| CHEMBL379975 | — | IC50 | = | 18086.27 | nM | 4.74 |
| CHEMBL573107 | — | IC50 | = | 18788.93 | nM | 4.73 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 21251.49 | nM | 4.67 |
| CHEMBL939 | GEFITINIB | IC50 | = | 22011.9 | nM | 4.66 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 22543.12 | nM | 4.65 |
| CHEMBL222102 | KU-55933 | IC50 | = | 25093.83 | nM | 4.60 |
| CHEMBL105442 | CI-1040 | IC50 | = | 25810.34 | nM | 4.59 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 28013.77 | nM | 4.55 |
| CHEMBL202721 | — | IC50 | = | 28635.64 | nM | 4.54 |