Assay Detail
Functional
CHEMBL2363693
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SANGER: Inhibition of human SW900 cell growth in a cell viability assay.
58
Total Activities
58
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SW900 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 58 | 5.26 | 8.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.12 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.59 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.50 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.21 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.81 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.61 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 5.97 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.95 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.85 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 5.79 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.76 |
| CHEMBL217354 | — | — | 1 | 5.56 |
| CHEMBL2137530 | SERDEMETAN | 2.0 | 1 | 5.46 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.43 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.17 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.11 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 4.97 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 4.95 |
| CHEMBL577784 | BX-795 | — | 1 | 4.88 |
| CHEMBL379975 | — | — | 1 | 4.78 |
| CHEMBL191334 | NUTLIN-3 | — | 1 | 4.77 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 4.68 |
| CHEMBL11359 | CISPLATIN | 4.0 | 1 | 4.54 |
| CHEMBL189584 | PD-173074 | — | 1 | 4.46 |
| CHEMBL176544 | — | — | 1 | 4.41 |
| CHEMBL188678 | — | — | 1 | 4.36 |
| CHEMBL399530 | — | — | 1 | 4.29 |
| CHEMBL572881 | MOTESANIB | 3.0 | 1 | 4.25 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 4.21 |
| CHEMBL202721 | — | — | 1 | 4.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 7.55 | nM | 8.12 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 25.41 | nM | 7.59 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 31.84 | nM | 7.50 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 62.12 | nM | 7.21 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 154.65 | nM | 6.81 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 245.79 | nM | 6.61 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 1078.3 | nM | 5.97 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 1122.51 | nM | 5.95 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1409.31 | nM | 5.85 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1621.61 | nM | 5.79 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1749.93 | nM | 5.76 |
| CHEMBL217354 | — | IC50 | = | 2769.86 | nM | 5.56 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 3482.55 | nM | 5.46 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 3721.51 | nM | 5.43 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 6762.21 | nM | 5.17 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 7821.21 | nM | 5.11 |
| CHEMBL939 | GEFITINIB | IC50 | = | 10822.81 | nM | 4.97 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 11239.92 | nM | 4.95 |
| CHEMBL577784 | BX-795 | IC50 | = | 13150.66 | nM | 4.88 |
| CHEMBL379975 | — | IC50 | = | 16553.71 | nM | 4.78 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 16913.18 | nM | 4.77 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 21014.93 | nM | 4.68 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 28933.61 | nM | 4.54 |
| CHEMBL189584 | PD-173074 | IC50 | = | 34811.51 | nM | 4.46 |
| CHEMBL176544 | — | IC50 | = | 38565.88 | nM | 4.41 |
| CHEMBL188678 | — | IC50 | = | 44075.76 | nM | 4.36 |
| CHEMBL399530 | — | IC50 | = | 51197.57 | nM | 4.29 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 55611.83 | nM | 4.25 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 61438.4 | nM | 4.21 |
| CHEMBL202721 | — | IC50 | = | 64654.58 | nM | 4.19 |
| CHEMBL105442 | CI-1040 | IC50 | = | 66377.89 | nM | 4.18 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 74983.12 | nM | 4.12 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 79655.89 | nM | 4.10 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 87205.29 | nM | 4.06 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 89816.8 | nM | 4.05 |
| CHEMBL102714 | SB-216763 | IC50 | = | 340331.11 | nM | - |
| CHEMBL506871 | VELIPARIB | IC50 | = | 256158.91 | nM | - |
| CHEMBL240954 | — | IC50 | = | 106553.37 | nM | - |
| CHEMBL3349342 | — | IC50 | = | 224904.3 | nM | - |
| CHEMBL477989 | SB590885 | IC50 | = | 277629.36 | nM | - |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 171743.14 | nM | - |
| CHEMBL255342 | — | IC50 | = | 798667.73 | nM | - |
| CHEMBL1186585 | — | IC50 | = | 2104813.2 | nM | - |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 300109.08 | nM | - |
| CHEMBL2134202 | — | IC50 | = | 198311.89 | nM | - |
| CHEMBL255863 | NILOTINIB | IC50 | = | 159446.59 | nM | - |
| CHEMBL38 | TRETINOIN | IC50 | = | 188385.43 | nM | - |
| CHEMBL483849 | — | IC50 | = | 4591417.14 | nM | - |
| CHEMBL1431 | METFORMIN | IC50 | = | 19285388.2 | nM | - |
| CHEMBL521686 | OLAPARIB | IC50 | = | 405371.93 | nM | - |