Assay Detail
Functional
CHEMBL2363700
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SANGER: Inhibition of human T-24 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T-24 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.56 | 8.81 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.81 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.79 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.29 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.91 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.86 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.77 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.71 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.68 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.36 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.27 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.11 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.78 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.61 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.61 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.55 |
| CHEMBL217354 | — | — | 1 | 6.53 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.48 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.43 |
| CHEMBL176544 | — | — | 1 | 6.20 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.14 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.11 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 5.72 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 5.68 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.65 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.61 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 5.61 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 5.61 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.58 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 5.54 |
| CHEMBL585951 | — | — | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1.551 | nM | 8.81 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.614 | nM | 8.79 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.104 | nM | 8.29 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 12.27 | nM | 7.91 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 13.86 | nM | 7.86 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 17.05 | nM | 7.77 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 19.71 | nM | 7.71 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 20.65 | nM | 7.68 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 43.83 | nM | 7.36 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 53.84 | nM | 7.27 |
| CHEMBL803 | CYTARABINE | IC50 | = | 78.56 | nM | 7.11 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 165.13 | nM | 6.78 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 245.77 | nM | 6.61 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 245.48 | nM | 6.61 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 284.25 | nM | 6.55 |
| CHEMBL217354 | — | IC50 | = | 294.56 | nM | 6.53 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 331.59 | nM | 6.48 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 369.85 | nM | 6.43 |
| CHEMBL176544 | — | IC50 | = | 638.23 | nM | 6.20 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 719.91 | nM | 6.14 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 778.71 | nM | 6.11 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1918.93 | nM | 5.72 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 2076.29 | nM | 5.68 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2255.44 | nM | 5.65 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 2478.81 | nM | 5.61 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 2480.37 | nM | 5.61 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 2462.32 | nM | 5.61 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 2600.62 | nM | 5.58 |
| CHEMBL105442 | CI-1040 | IC50 | = | 2911.12 | nM | 5.54 |
| CHEMBL585951 | — | IC50 | = | 2868.97 | nM | 5.54 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3150.7 | nM | 5.50 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 3218.14 | nM | 5.49 |
| CHEMBL379975 | — | IC50 | = | 4935.3 | nM | 5.31 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 5561.56 | nM | 5.25 |
| CHEMBL135561 | — | IC50 | = | 6329.47 | nM | 5.20 |
| CHEMBL103667 | DORAMAPIMOD | IC50 | = | 8406.73 | nM | 5.08 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 9658.07 | nM | 5.01 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 9688.15 | nM | 5.01 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 9944.15 | nM | 5.00 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 10940.35 | nM | 4.96 |
| CHEMBL399530 | — | IC50 | = | 13153.75 | nM | 4.88 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 13915.66 | nM | 4.86 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 13954.82 | nM | 4.86 |
| CHEMBL202721 | — | IC50 | = | 15254.6 | nM | 4.82 |
| CHEMBL577784 | BX-795 | IC50 | = | 16297.83 | nM | 4.79 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 17534.69 | nM | 4.76 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 18086.77 | nM | 4.74 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 18692.49 | nM | 4.73 |
| CHEMBL1190711 | — | IC50 | = | 22715.78 | nM | 4.64 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 28192.5 | nM | 4.55 |