Assay Detail
Functional
CHEMBL2363701
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SANGER: Inhibition of human T47D cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T47D |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.22 | 8.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.37 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.11 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.87 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.78 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.17 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.97 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.82 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.65 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 6.56 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.56 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.55 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.40 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 6.35 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.33 |
| CHEMBL258844 | — | — | 1 | 6.29 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 6.27 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.22 |
| CHEMBL217354 | — | — | 1 | 6.16 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.91 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.78 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 5.64 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 5.51 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.49 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 5.44 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.32 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 5.28 |
| CHEMBL573107 | — | — | 1 | 5.22 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.20 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.20 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 4.309 | nM | 8.37 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 7.711 | nM | 8.11 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 13.52 | nM | 7.87 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 16.79 | nM | 7.78 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 67.87 | nM | 7.17 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 107.46 | nM | 6.97 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 152.98 | nM | 6.82 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 223.06 | nM | 6.65 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 278.17 | nM | 6.56 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 274.75 | nM | 6.56 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 282.5 | nM | 6.55 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 400.41 | nM | 6.40 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 445.28 | nM | 6.35 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 469.69 | nM | 6.33 |
| CHEMBL258844 | — | IC50 | = | 516.2 | nM | 6.29 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 532.7 | nM | 6.27 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 597.56 | nM | 6.22 |
| CHEMBL217354 | — | IC50 | = | 690.67 | nM | 6.16 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 937.97 | nM | 6.03 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1236.96 | nM | 5.91 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1680.61 | nM | 5.78 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 2279.99 | nM | 5.64 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 3105.58 | nM | 5.51 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3236.27 | nM | 5.49 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 3622.17 | nM | 5.44 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 4766.35 | nM | 5.32 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 5248.03 | nM | 5.28 |
| CHEMBL573107 | — | IC50 | = | 5961.2 | nM | 5.22 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 6264.57 | nM | 5.20 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 6371.91 | nM | 5.20 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 7000.94 | nM | 5.16 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 8160.24 | nM | 5.09 |
| CHEMBL176544 | — | IC50 | = | 9207.99 | nM | 5.04 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 10154.98 | nM | 4.99 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 11663.66 | nM | 4.93 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 12258.04 | nM | 4.91 |
| CHEMBL848 | LENALIDOMIDE | IC50 | = | 13209.85 | nM | 4.88 |
| CHEMBL1186585 | — | IC50 | = | 14649.88 | nM | 4.83 |
| CHEMBL585951 | — | IC50 | = | 17549.67 | nM | 4.76 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 18220.18 | nM | 4.74 |
| CHEMBL188678 | — | IC50 | = | 18487.98 | nM | 4.73 |
| CHEMBL2134202 | — | IC50 | = | 20148.5 | nM | 4.70 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 20927.12 | nM | 4.68 |
| CHEMBL1090090 | VX-702 | IC50 | = | 21224.26 | nM | 4.67 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 21787.62 | nM | 4.66 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 22797.94 | nM | 4.64 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 24878.35 | nM | 4.60 |
| CHEMBL202721 | — | IC50 | = | 25509.27 | nM | 4.59 |
| CHEMBL255342 | — | IC50 | = | 25513.2 | nM | 4.59 |
| CHEMBL2363137 | — | IC50 | = | 26919.85 | nM | 4.57 |