Assay Detail
Functional
CHEMBL2363721
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SANGER: Inhibition of human A204 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A204 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.90 | 8.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.51 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.49 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.34 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 8.07 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.06 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.05 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.03 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 8.00 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.95 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 7.91 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.89 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.76 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.67 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.65 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.55 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.41 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.08 |
| CHEMBL217354 | — | — | 1 | 7.01 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 7.00 |
| CHEMBL477772 | PAZOPANIB | 4.0 | 1 | 6.96 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.90 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.82 |
| CHEMBL585951 | — | — | 1 | 6.78 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.72 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.70 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.65 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.63 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.51 |
| CHEMBL572881 | MOTESANIB | 3.0 | 1 | 6.29 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 3.12 | nM | 8.51 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.208 | nM | 8.49 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 4.525 | nM | 8.34 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 8.562 | nM | 8.07 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 8.765 | nM | 8.06 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 8.848 | nM | 8.05 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 9.339 | nM | 8.03 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 9.923 | nM | 8.00 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 11.16 | nM | 7.95 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 12.18 | nM | 7.91 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 12.88 | nM | 7.89 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 17.29 | nM | 7.76 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 21.15 | nM | 7.67 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 22.49 | nM | 7.65 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 28.47 | nM | 7.55 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 38.85 | nM | 7.41 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 84.19 | nM | 7.08 |
| CHEMBL217354 | — | IC50 | = | 97.84 | nM | 7.01 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 100.52 | nM | 7.00 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 109.06 | nM | 6.96 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 126.54 | nM | 6.90 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 151.59 | nM | 6.82 |
| CHEMBL585951 | — | IC50 | = | 164.53 | nM | 6.78 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 189.7 | nM | 6.72 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 200.37 | nM | 6.70 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 221.9 | nM | 6.65 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 232.48 | nM | 6.63 |
| CHEMBL803 | CYTARABINE | IC50 | = | 310.68 | nM | 6.51 |
| CHEMBL572881 | MOTESANIB | IC50 | = | 518.54 | nM | 6.29 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 522.33 | nM | 6.28 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 633.91 | nM | 6.20 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 1084.08 | nM | 5.96 |
| CHEMBL577784 | BX-795 | IC50 | = | 1154.67 | nM | 5.94 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1516.67 | nM | 5.82 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1598.01 | nM | 5.80 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 1572.05 | nM | 5.80 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1770.17 | nM | 5.75 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 2483.96 | nM | 5.61 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 2767.32 | nM | 5.56 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 2838.72 | nM | 5.55 |
| CHEMBL191334 | NUTLIN-3 | IC50 | = | 3055.88 | nM | 5.51 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 3580.82 | nM | 5.45 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 3909.56 | nM | 5.41 |
| CHEMBL189584 | PD-173074 | IC50 | = | 3920.75 | nM | 5.41 |
| CHEMBL202721 | — | IC50 | = | 4394.08 | nM | 5.36 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 4358.03 | nM | 5.36 |
| CHEMBL379975 | — | IC50 | = | 4466.38 | nM | 5.35 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 5306.92 | nM | 5.28 |
| CHEMBL2363137 | — | IC50 | = | 6086.52 | nM | 5.22 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 7064.72 | nM | 5.15 |