Assay Detail
ADMET
CHEMBL2390496
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Cytotoxicity against rat L6 cells after 72 hrs by Alamar blue assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Rattus norvegicus |
| Cell Type | L6 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
New Promising Compounds with in Vitro Nanomolar Activity against Trypanosoma cruzi.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.03 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 9.00 |
| CHEMBL1946928 | — | — | 1 | 4.89 |
| CHEMBL2385091 | — | — | 1 | 4.87 |
| CHEMBL2386136 | — | — | 1 | 4.86 |
| CHEMBL2386137 | — | — | 1 | 4.81 |
| CHEMBL1946927 | — | — | 1 | 4.78 |
| CHEMBL2386135 | — | — | 1 | 4.74 |
| CHEMBL1946738 | — | — | 1 | 4.63 |
| CHEMBL1946929 | — | — | 1 | 4.57 |
| CHEMBL2386134 | — | — | 1 | 4.56 |
| CHEMBL2386138 | — | — | 1 | 4.50 |
| CHEMBL2386132 | — | — | 1 | 4.10 |
| CHEMBL2386133 | — | — | 1 | - |
| CHEMBL2386131 | — | — | 1 | - |
| CHEMBL1946741 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL61 | PODOFILOX | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1946928 | — | IC50 | = | 12970.0 | nM | 4.89 |
| CHEMBL2385091 | — | IC50 | = | 13440.0 | nM | 4.87 |
| CHEMBL2386136 | — | IC50 | = | 13960.0 | nM | 4.86 |
| CHEMBL2386137 | — | IC50 | = | 15380.0 | nM | 4.81 |
| CHEMBL1946927 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL2386135 | — | IC50 | = | 18240.0 | nM | 4.74 |
| CHEMBL1946738 | — | IC50 | = | 23590.0 | nM | 4.63 |
| CHEMBL1946929 | — | IC50 | = | 27200.0 | nM | 4.57 |
| CHEMBL2386134 | — | IC50 | = | 27500.0 | nM | 4.56 |
| CHEMBL2386138 | — | IC50 | = | 31560.0 | nM | 4.50 |
| CHEMBL2386132 | — | IC50 | = | 79300.0 | nM | 4.10 |
| CHEMBL2386133 | — | IC50 | = | 237600.0 | nM | - |
| CHEMBL2386131 | — | IC50 | = | 222100.0 | nM | - |
| CHEMBL1946741 | — | IC50 | = | 182500.0 | nM | - |