Assay Detail
Binding
CHEMBL2399175
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Binding affinity to mu opioid receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Orally active opioid compounds from a non-poppy source.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.58 | 11.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL58362 | — | — | 1 | 11.00 |
| CHEMBL2396991 | — | — | 1 | 8.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL58362 | — | Ki | = | 0.01 | nM | 11.00 |
| CHEMBL2396991 | — | Ki | = | 7.0 | nM | 8.15 |