Assay Detail
Functional
CHEMBL2445704
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human ECV304 cells after 72 hrs by MTT assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | ECV-304 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
The influence of saponins on cell membrane cholesterol.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 4.67 | 5.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2442199 | — | — | 1 | 5.10 |
| CHEMBL2442201 | — | — | 1 | 5.05 |
| CHEMBL2442200 | — | — | 1 | 4.89 |
| CHEMBL447565 | ALPHA-HEDERIN | — | 1 | 4.46 |
| CHEMBL504794 | beta-ESCIN | — | 1 | 4.28 |
| CHEMBL221542 | BETA-SITOSTEROL | — | 1 | 4.21 |
| CHEMBL2442203 | — | — | 1 | - |
| CHEMBL2442202 | — | — | 1 | - |
| CHEMBL1910840 | KALOPANAXSAPONIN B | — | 1 | - |
| CHEMBL441687 | GLYCYRRHIZIN | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2442199 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL2442201 | — | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL2442200 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL447565 | ALPHA-HEDERIN | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL504794 | beta-ESCIN | IC50 | = | 52000.0 | nM | 4.28 |
| CHEMBL221542 | BETA-SITOSTEROL | IC50 | = | 61000.0 | nM | 4.21 |
| CHEMBL2442203 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2442202 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1910840 | KALOPANAXSAPONIN B | IC50 | > | 164000.0 | nM | - |
| CHEMBL441687 | GLYCYRRHIZIN | IC50 | > | 119000.0 | nM | - |