Assay Detail
Binding
CHEMBL3215092
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Counterscreen for inhibitors of LEDGF/p75-dependent integration: TR-FRET-based biochemical high throughput dose response counterscreen assay to identify activators of HIV-1 Integrase multimerization. (Class of assay: confirmatory)
239
Total Activities
239
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 239 | 5.16 | 7.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1986342 | — | — | 1 | 7.07 |
| CHEMBL1329826 | — | — | 1 | 7.04 |
| CHEMBL1302308 | — | — | 1 | 6.71 |
| CHEMBL1468796 | — | — | 1 | 6.61 |
| CHEMBL1723511 | — | — | 1 | 6.46 |
| CHEMBL1601846 | — | — | 1 | 6.45 |
| CHEMBL3191022 | — | — | 1 | 6.25 |
| CHEMBL1503050 | — | — | 1 | 6.17 |
| CHEMBL1541 | CEFIXIME | 4.0 | 1 | 6.12 |
| CHEMBL1362935 | — | — | 1 | 6.08 |
| CHEMBL1407474 | — | — | 1 | 6.06 |
| CHEMBL1730974 | — | — | 1 | 6.02 |
| CHEMBL164 | MYRICETIN | — | 1 | 5.94 |
| CHEMBL3197557 | — | — | 1 | 5.89 |
| CHEMBL1484234 | — | — | 1 | 5.88 |
| CHEMBL1700996 | — | — | 1 | 5.87 |
| CHEMBL1373655 | — | — | 1 | 5.85 |
| CHEMBL1728023 | — | — | 1 | 5.84 |
| CHEMBL1727349 | — | — | 1 | 5.81 |
| CHEMBL175266 | — | — | 1 | 5.81 |
| CHEMBL1735454 | — | — | 1 | 5.80 |
| CHEMBL1718398 | — | — | 1 | 5.73 |
| CHEMBL1533230 | — | — | 1 | 5.72 |
| CHEMBL405110 | METHYLENE BLUE ANHYDROUS | 4.0 | 1 | 5.71 |
| CHEMBL1301673 | — | — | 1 | 5.67 |
| CHEMBL3194876 | — | — | 1 | 5.65 |
| CHEMBL1706454 | — | — | 1 | 5.64 |
| CHEMBL1320230 | — | — | 1 | 5.61 |
| CHEMBL1985664 | — | — | 1 | 5.60 |
| CHEMBL1385808 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1986342 | — | IC50 | = | 84.96 | nM | 7.07 |
| CHEMBL1329826 | — | IC50 | = | 92.27 | nM | 7.04 |
| CHEMBL1302308 | — | IC50 | = | 196.73 | nM | 6.71 |
| CHEMBL1468796 | — | IC50 | = | 245.27 | nM | 6.61 |
| CHEMBL1723511 | — | IC50 | = | 347.95 | nM | 6.46 |
| CHEMBL1601846 | — | IC50 | = | 353.89 | nM | 6.45 |
| CHEMBL3191022 | — | IC50 | = | 563.94 | nM | 6.25 |
| CHEMBL1503050 | — | IC50 | = | 676.63 | nM | 6.17 |
| CHEMBL1541 | CEFIXIME | IC50 | = | 759.02 | nM | 6.12 |
| CHEMBL1362935 | — | IC50 | = | 833.7 | nM | 6.08 |
| CHEMBL1407474 | — | IC50 | = | 869.51 | nM | 6.06 |
| CHEMBL1730974 | — | IC50 | = | 953.0 | nM | 6.02 |
| CHEMBL164 | MYRICETIN | IC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL3197557 | — | IC50 | = | 1288.0 | nM | 5.89 |
| CHEMBL1484234 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1700996 | — | IC50 | = | 1351.0 | nM | 5.87 |
| CHEMBL1373655 | — | IC50 | = | 1414.0 | nM | 5.85 |
| CHEMBL1728023 | — | IC50 | = | 1449.0 | nM | 5.84 |
| CHEMBL175266 | — | IC50 | = | 1536.0 | nM | 5.81 |
| CHEMBL1727349 | — | IC50 | = | 1563.0 | nM | 5.81 |
| CHEMBL1735454 | — | IC50 | = | 1568.0 | nM | 5.80 |
| CHEMBL1718398 | — | IC50 | = | 1874.0 | nM | 5.73 |
| CHEMBL1533230 | — | IC50 | = | 1921.0 | nM | 5.72 |
| CHEMBL405110 | METHYLENE BLUE ANHYDROUS | IC50 | = | 1958.0 | nM | 5.71 |
| CHEMBL1301673 | — | IC50 | = | 2130.0 | nM | 5.67 |
| CHEMBL3194876 | — | IC50 | = | 2223.0 | nM | 5.65 |
| CHEMBL1706454 | — | IC50 | = | 2299.0 | nM | 5.64 |
| CHEMBL1320230 | — | IC50 | = | 2454.0 | nM | 5.61 |
| CHEMBL1985664 | — | IC50 | = | 2497.0 | nM | 5.60 |
| CHEMBL1385808 | — | IC50 | = | 2533.0 | nM | 5.60 |
| CHEMBL1601394 | — | IC50 | = | 2619.0 | nM | 5.58 |
| CHEMBL1488474 | — | IC50 | = | 2654.0 | nM | 5.58 |
| CHEMBL1323674 | — | IC50 | = | 2717.0 | nM | 5.57 |
| CHEMBL1713097 | — | IC50 | = | 2858.0 | nM | 5.54 |
| CHEMBL1567396 | — | IC50 | = | 3015.0 | nM | 5.52 |
| CHEMBL1968928 | — | IC50 | = | 3010.0 | nM | 5.52 |
| CHEMBL1508847 | — | IC50 | = | 3309.0 | nM | 5.48 |
| CHEMBL1972037 | — | IC50 | = | 3401.0 | nM | 5.47 |
| CHEMBL1419228 | — | IC50 | = | 3567.0 | nM | 5.45 |
| CHEMBL515252 | — | IC50 | = | 3520.0 | nM | 5.45 |
| CHEMBL1271266 | — | IC50 | = | 3590.0 | nM | 5.45 |
| CHEMBL1708760 | — | IC50 | = | 3564.0 | nM | 5.45 |
| CHEMBL1493010 | — | IC50 | = | 3645.0 | nM | 5.44 |
| CHEMBL3196993 | — | IC50 | = | 3717.0 | nM | 5.43 |
| CHEMBL1966984 | — | IC50 | = | 3759.0 | nM | 5.42 |
| CHEMBL3191780 | — | IC50 | = | 3861.0 | nM | 5.41 |
| CHEMBL1555751 | — | IC50 | = | 3896.0 | nM | 5.41 |
| CHEMBL1429070 | — | IC50 | = | 4005.0 | nM | 5.40 |
| CHEMBL1424694 | — | IC50 | = | 4170.0 | nM | 5.38 |
| CHEMBL290914 | EMODIC ACID | IC50 | = | 4190.0 | nM | 5.38 |