Assay Detail
Binding
CHEMBL3268708
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Inhibition of Syk (unknown origin) using 4 uM peptide assessed as product formation after 60 mins incubation by microfluidic mobility shift assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Syk inhibitors with high potency in presence of blood.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 7.75 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3262620 | — | — | 1 | 9.00 |
| CHEMBL3262622 | — | — | 1 | 9.00 |
| CHEMBL3262616 | — | — | 1 | 9.00 |
| CHEMBL3262357 | — | — | 1 | 8.70 |
| CHEMBL3262625 | — | — | 1 | 8.52 |
| CHEMBL3262356 | — | — | 1 | 8.40 |
| CHEMBL3262623 | — | — | 1 | 8.40 |
| CHEMBL3262355 | — | — | 1 | 8.30 |
| CHEMBL2177736 | — | — | 1 | 7.89 |
| CHEMBL3262617 | — | — | 1 | 7.70 |
| CHEMBL3262618 | — | — | 1 | 7.68 |
| CHEMBL3262624 | — | — | 1 | 7.66 |
| CHEMBL3262358 | — | — | 1 | 7.47 |
| CHEMBL475251 | R-406 | 2.0 | 1 | 7.17 |
| CHEMBL3262619 | — | — | 1 | 6.78 |
| CHEMBL3262621 | — | — | 1 | 6.32 |
| CHEMBL3262359 | — | — | 1 | 5.80 |
| CHEMBL3262626 | — | — | 1 | 5.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3262620 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3262622 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3262616 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3262357 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3262625 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3262356 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3262623 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3262355 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL2177736 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL3262617 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3262618 | — | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL3262624 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL3262358 | — | IC50 | = | 34.0 | nM | 7.47 |
| CHEMBL475251 | R-406 | IC50 | = | 68.0 | nM | 7.17 |
| CHEMBL3262619 | — | IC50 | = | 165.0 | nM | 6.78 |
| CHEMBL3262621 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL3262359 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL3262626 | — | IC50 | = | 1900.0 | nM | 5.72 |