Assay Detail
Functional
CHEMBL3268712
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Inhibition of IL3 dependent proliferation in C57/B16 mouse bone marrow cells using [3H]thymidine by liquid scintillation counting
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | Bone marrow cell |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Syk inhibitors with high potency in presence of blood.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 5.59 | 6.83 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL475251 | R-406 | 2.0 | 1 | 6.83 |
| CHEMBL3262355 | — | — | 1 | 6.60 |
| CHEMBL3262622 | — | — | 1 | 5.84 |
| CHEMBL3262356 | — | — | 1 | 5.47 |
| CHEMBL3262624 | — | — | 1 | 5.45 |
| CHEMBL3262357 | — | — | 1 | 5.42 |
| CHEMBL3262616 | — | — | 1 | 5.38 |
| CHEMBL3262625 | — | — | 1 | 5.31 |
| CHEMBL2177736 | — | — | 1 | 5.23 |
| CHEMBL3262620 | — | — | 1 | 5.22 |
| CHEMBL3262358 | — | — | 1 | 5.18 |
| CHEMBL3262617 | — | — | 1 | 5.13 |
| CHEMBL3262618 | — | — | 1 | - |
| CHEMBL3262619 | — | — | 1 | - |
| CHEMBL3262621 | — | — | 1 | - |
| CHEMBL3262359 | — | — | 1 | - |
| CHEMBL3262623 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL475251 | R-406 | IC50 | = | 147.0 | nM | 6.83 |
| CHEMBL3262355 | — | IC50 | = | 249.0 | nM | 6.60 |
| CHEMBL3262622 | — | IC50 | = | 1443.0 | nM | 5.84 |
| CHEMBL3262356 | — | IC50 | = | 3411.0 | nM | 5.47 |
| CHEMBL3262624 | — | IC50 | = | 3514.0 | nM | 5.45 |
| CHEMBL3262357 | — | IC50 | = | 3796.0 | nM | 5.42 |
| CHEMBL3262616 | — | IC50 | = | 4139.0 | nM | 5.38 |
| CHEMBL3262625 | — | IC50 | = | 4938.0 | nM | 5.31 |
| CHEMBL2177736 | — | IC50 | = | 5853.0 | nM | 5.23 |
| CHEMBL3262620 | — | IC50 | = | 5984.0 | nM | 5.22 |
| CHEMBL3262358 | — | IC50 | = | 6664.0 | nM | 5.18 |
| CHEMBL3262617 | — | IC50 | = | 7474.0 | nM | 5.13 |
| CHEMBL3262618 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3262619 | — | IC50 | - | — | - | |
| CHEMBL3262621 | — | IC50 | - | — | - | |
| CHEMBL3262359 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3262623 | — | IC50 | - | — | - |