Assay Detail
Functional
CHEMBL3363331
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Inhibition of FMLP/CB-stimulated superoxide production in human neutrophils preincubated for 5 mins before FMLP/CB treatment by spectrophotometry
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Neutrophil |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Anti-Inflammatory Spirostanol and Furostanol Saponins from Solanum macaonense.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.40 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL365739 | DIPHENYLENEIODONIUM | — | 1 | 6.10 |
| CHEMBL504101 | — | — | 1 | 5.40 |
| CHEMBL2047364 | CHLOROGENIN | — | 1 | 5.21 |
| CHEMBL505565 | — | — | 1 | 5.16 |
| CHEMBL466034 | — | — | 1 | 5.12 |
| CHEMBL3329787 | — | — | 1 | - |
| CHEMBL3329788 | — | — | 1 | - |
| CHEMBL3329789 | — | — | 1 | - |
| CHEMBL3329790 | — | — | 1 | - |
| CHEMBL3329786 | — | — | 1 | - |
| CHEMBL3329792 | — | — | 1 | - |
| CHEMBL3329793 | — | — | 1 | - |
| CHEMBL3329794 | — | — | 1 | - |
| CHEMBL3329795 | — | — | 1 | - |
| CHEMBL3329796 | — | — | 1 | - |
| CHEMBL3329797 | — | — | 1 | - |
| CHEMBL3329798 | — | — | 1 | - |
| CHEMBL3329799 | — | — | 1 | - |
| CHEMBL3329800 | — | — | 1 | - |
| CHEMBL3331544 | — | — | 1 | - |
| CHEMBL3329791 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL365739 | DIPHENYLENEIODONIUM | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL504101 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL2047364 | CHLOROGENIN | IC50 | = | 6100.0 | nM | 5.21 |
| CHEMBL505565 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL466034 | — | IC50 | = | 7600.0 | nM | 5.12 |
| CHEMBL3329787 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329788 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329789 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329790 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329786 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329792 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329793 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329794 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329795 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329796 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329797 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329798 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329799 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329800 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3331544 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3329791 | — | IC50 | > | 10000.0 | nM | - |