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Compound Detail

CHEMBL2047364

CHLOROGENIN
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C[C@@H]1CC[C@@]2(OC1)O[C@H]1C[C@H]3[C@@H]4C[C@H](O)[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]1[C@@H]2C

Basic Information

ChEMBL ID CHEMBL2047364
Name CHLOROGENIN
Phase Preclinical
Structure Type MOL
InChI Key PZNPHSFXILSZTM-JUGSJECZSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

432.6
MW (Da)
4.76
ALogP
4
HBA
2
HBD
58.9
PSA (Ų)
0.58
QED
0
Ro5 Violations
0
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C27H44O4
MW 432.65
Aromatic Rings 0
Heavy Atoms 31
NP-Likeness 3.21

Activity Summary

IC50 1 meas. best 5.21

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Neutrophil
CHEMBL613710
IC50 5.21 5.21 6100.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Neutrophil IC50 = 6100.0 nM 5.21 Inhibition of FMLP/CB-stimulated superoxide production in human neutrophils prei... 25036668

Literature References

PubMed DOI Target Context # Activities
22575533 10.1016/j.ejmech.2012.04.022 NON-PROTEIN TARGET 2
25036668 10.1021/np500057b Neutrophil 2

Data from ChEMBL 36 via Core Engine