Assay Detail
Functional
CHEMBL3384520
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human MIAPaCa2 cells after 24 hrs by WST-1 assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MIA PaCa-2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Tailor-made fluorescent trilobolide to study its biological relevance.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 4.76 | 4.76 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3343188 | — | — | 1 | 4.76 |
| CHEMBL3343189 | — | — | 1 | - |
| CHEMBL3343190 | — | — | 1 | - |
| CHEMBL3343191 | — | — | 1 | - |
| CHEMBL3343192 | — | — | 1 | - |
| CHEMBL3343405 | — | — | 1 | - |
| CHEMBL3343406 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3343188 | — | IC50 | = | 17400.0 | nM | 4.76 |
| CHEMBL3343189 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3343190 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3343191 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3343192 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3343405 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL3343406 | — | IC50 | > | 50000.0 | nM | - |