Assay Detail
Binding
CHEMBL3395903
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Inhibition of p38 (unknown origin)
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Inhibitors of c-Jun N-terminal kinases: an update.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 6.48 | 7.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1233748 | — | — | 1 | 7.52 |
| CHEMBL1233747 | — | — | 1 | 5.43 |
| CHEMBL3393599 | — | — | 1 | - |
| CHEMBL571626 | — | — | 1 | - |
| CHEMBL585951 | — | — | 1 | - |
| CHEMBL2144409 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1233748 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL1233747 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL3393599 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL571626 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL585951 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL2144409 | — | IC50 | > | 20000.0 | nM | - |