Assay Detail
Functional
CHEMBL3413799
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Respiratory syncytial virus A2 infected in human Hep2 cells assessed as protection against virus-induced cytopathogenicity after 4 days by cell-Titer Glo assay
42
Total Activities
42
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Respiratory syncytial virus |
| Cell Type | HEp-2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Respiratory syncytial virus (CHEMBL612679) ↗| Type | ORGANISM |
| Organism | Respiratory syncytial virus |
Publication
Discovery of an oral respiratory syncytial virus (RSV) fusion inhibitor (GS-5806) and clinical proof of concept in a human RSV challenge study.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 42 | 7.65 | 9.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3410450 | PRESATOVIR | 2.0 | 1 | 9.43 |
| CHEMBL3410445 | — | — | 1 | 9.19 |
| CHEMBL3410446 | — | — | 1 | 9.14 |
| CHEMBL3410438 | — | — | 1 | 8.96 |
| CHEMBL3410435 | — | — | 1 | 8.92 |
| CHEMBL3410442 | — | — | 1 | 8.82 |
| CHEMBL3410441 | — | — | 1 | 8.82 |
| CHEMBL3410436 | — | — | 1 | 8.68 |
| CHEMBL3410449 | — | — | 1 | 8.59 |
| CHEMBL3410439 | — | — | 1 | 8.52 |
| CHEMBL3410443 | — | — | 1 | 8.36 |
| CHEMBL3410447 | — | — | 1 | 8.35 |
| CHEMBL3410423 | — | — | 1 | 8.30 |
| CHEMBL3410444 | — | — | 1 | 8.27 |
| CHEMBL3410433 | — | — | 1 | 8.26 |
| CHEMBL3410437 | — | — | 1 | 8.15 |
| CHEMBL3410448 | — | — | 1 | 8.12 |
| CHEMBL3410432 | — | — | 1 | 8.12 |
| CHEMBL3410431 | — | — | 1 | 8.03 |
| CHEMBL3407530 | — | — | 1 | 7.85 |
| CHEMBL3410440 | — | — | 1 | 7.70 |
| CHEMBL3410434 | — | — | 1 | 7.64 |
| CHEMBL3410430 | — | — | 1 | 7.57 |
| CHEMBL3410425 | — | — | 1 | 7.54 |
| CHEMBL3410427 | — | — | 1 | 7.35 |
| CHEMBL3410429 | — | — | 1 | 7.31 |
| CHEMBL3410416 | — | — | 1 | 7.24 |
| CHEMBL3410412 | — | — | 1 | 7.19 |
| CHEMBL3410420 | — | — | 1 | 7.13 |
| CHEMBL3410422 | — | — | 1 | 7.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3410450 | PRESATOVIR | EC50 | = | 0.37 | nM | 9.43 |
| CHEMBL3410445 | — | EC50 | = | 0.64 | nM | 9.19 |
| CHEMBL3410446 | — | EC50 | = | 0.72 | nM | 9.14 |
| CHEMBL3410438 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL3410435 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL3410442 | — | EC50 | = | 1.5 | nM | 8.82 |
| CHEMBL3410441 | — | EC50 | = | 1.5 | nM | 8.82 |
| CHEMBL3410436 | — | EC50 | = | 2.1 | nM | 8.68 |
| CHEMBL3410449 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL3410439 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3410443 | — | EC50 | = | 4.4 | nM | 8.36 |
| CHEMBL3410447 | — | EC50 | = | 4.5 | nM | 8.35 |
| CHEMBL3410423 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL3410444 | — | EC50 | = | 5.4 | nM | 8.27 |
| CHEMBL3410433 | — | EC50 | = | 5.5 | nM | 8.26 |
| CHEMBL3410437 | — | EC50 | = | 7.0 | nM | 8.15 |
| CHEMBL3410448 | — | EC50 | = | 7.5 | nM | 8.12 |
| CHEMBL3410432 | — | EC50 | = | 7.5 | nM | 8.12 |
| CHEMBL3410431 | — | EC50 | = | 9.4 | nM | 8.03 |
| CHEMBL3407530 | — | EC50 | = | 14.0 | nM | 7.85 |
| CHEMBL3410440 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3410434 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL3410430 | — | EC50 | = | 27.0 | nM | 7.57 |
| CHEMBL3410425 | — | EC50 | = | 29.0 | nM | 7.54 |
| CHEMBL3410427 | — | EC50 | = | 45.0 | nM | 7.35 |
| CHEMBL3410429 | — | EC50 | = | 49.0 | nM | 7.31 |
| CHEMBL3410416 | — | EC50 | = | 57.0 | nM | 7.24 |
| CHEMBL3410412 | — | EC50 | = | 65.0 | nM | 7.19 |
| CHEMBL3410420 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL3410422 | — | EC50 | = | 81.0 | nM | 7.09 |
| CHEMBL3410428 | — | EC50 | = | 180.0 | nM | 6.75 |
| CHEMBL3410410 | — | EC50 | = | 202.0 | nM | 6.70 |
| CHEMBL3410417 | — | EC50 | = | 212.0 | nM | 6.67 |
| CHEMBL3410418 | — | EC50 | = | 305.0 | nM | 6.52 |
| CHEMBL3410415 | — | EC50 | = | 331.0 | nM | 6.48 |
| CHEMBL3410421 | — | EC50 | = | 402.0 | nM | 6.40 |
| CHEMBL3410419 | — | EC50 | = | 429.0 | nM | 6.37 |
| CHEMBL3410413 | — | EC50 | = | 586.0 | nM | 6.23 |
| CHEMBL3410414 | — | EC50 | = | 861.0 | nM | 6.07 |
| CHEMBL3410424 | — | EC50 | = | 2606.0 | nM | 5.58 |
| CHEMBL3410411 | — | EC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL3410426 | — | EC50 | > | 10000.0 | nM | - |