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Assay Detail

CHEMBL3420218

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of equine serum BuChE pre-incubated for 5 mins before butyrylthiocholine iodide substrate by Ellman' method
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Equus caballus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cholinesterase (CHEMBL5763)
Type SINGLE PROTEIN
Organism Equus caballus

Publication

Novel multitarget-directed ligands (MTDLs) with acetylcholinesterase (AChE) inhibitory and serotonergic subtype 4 receptor (5-HT4R) agonist activities as potential agents against Alzheimer's disease: the design of donecopride.
Rochais C, Lecoutey C, Gaven F, Giannoni P, Hamidouche K, Hedou D, Dubost E, Genest D, Yahiaoui S, Freret T, Bouet V, Dauphin F, Sopkova de Oliveira Santos J, Ballandonne C, Corvaisier S, Malzert-Fréon A, Legay R, Boulouard M, Claeysen S, Dallemagne P.
J Med Chem (2015) 58 : 3172 -3187
PubMed 25793650 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 14 5.29 5.74

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3417001 1 5.74
CHEMBL3417009 1 5.45
CHEMBL3417006 1 5.44
CHEMBL3416997 1 5.40
CHEMBL3417008 1 5.39
CHEMBL3417000 1 5.36
CHEMBL3416999 1 5.20
CHEMBL3414597 1 5.18
CHEMBL502 DONEPEZIL 4.0 1 5.16
CHEMBL3416996 1 5.16
CHEMBL3417004 1 5.15
CHEMBL3417005 1 5.13
CHEMBL3417002 1 5.04
CHEMBL3417007 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3417001 IC50 = 1835.0 nM 5.74
CHEMBL3417009 IC50 = 3530.0 nM 5.45
CHEMBL3417006 IC50 = 3640.0 nM 5.44
CHEMBL3416997 IC50 = 4000.0 nM 5.40
CHEMBL3417008 IC50 = 4100.0 nM 5.39
CHEMBL3417000 IC50 = 4340.0 nM 5.36
CHEMBL3416999 IC50 = 6340.0 nM 5.20
CHEMBL3414597 IC50 = 6600.0 nM 5.18
CHEMBL502 DONEPEZIL IC50 = 7000.0 nM 5.16
CHEMBL3416996 IC50 = 6910.0 nM 5.16
CHEMBL3417004 IC50 = 7080.0 nM 5.15
CHEMBL3417005 IC50 = 7420.0 nM 5.13
CHEMBL3417002 IC50 = 9165.0 nM 5.04
CHEMBL3417007 IC50 - -