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Assay Detail

CHEMBL3423893

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of human recombinant CYP2A6 assessed as metabolism of coumarin to 7-hydroxycoumarin after 30 mins by fluorescence assay
4
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 2A6 (CHEMBL5282)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design and synthesis of norendoxifen analogues with dual aromatase inhibitory and estrogen receptor modulatory activities.
Lv W, Liu J, Skaar TC, Flockhart DA, Cushman M.
J Med Chem (2015) 58 : 2623 -2648
PubMed 25751283 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.20 5.20
Ki 2 5.91 6.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3422028 2 6.15
CHEMBL2386285 2 5.66

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3422028 Ki = 710.0 nM 6.15
CHEMBL2386285 Ki = 2180.0 nM 5.66
CHEMBL2386285 IC50 = 6370.0 nM 5.20
CHEMBL3422028 IC50 = 6370.0 nM 5.20