Assay Detail
Functional
CHEMBL3562043
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. VEGF stimulated ADSC/ECFC co-culture CD31-stained tube area decrease-IC50. (Class of assay: confirmatory)
369
Total Activities
368
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 369 | 6.16 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.00 |
| CHEMBL1554 | DACTINOMYCIN | 4.0 | 1 | 9.00 |
| CHEMBL1289926 | AXITINIB | 4.0 | 1 | 8.89 |
| CHEMBL113051 | GIMATECAN | 2.0 | 1 | 8.70 |
| CHEMBL378544 | VINBLASTINE SULFATE | 4.0 | 2 | 8.64 |
| CHEMBL3182961 | — | — | 1 | 8.52 |
| CHEMBL3559830 | — | — | 1 | 8.39 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | 4.0 | 1 | 8.36 |
| CHEMBL538943 | VINORELBINE TARTRATE | 4.0 | 1 | 8.26 |
| CHEMBL2354444 | PIRARUBICIN | 3.0 | 1 | 8.20 |
| CHEMBL90555 | VINCRISTINE | 4.0 | 1 | 8.19 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 8.09 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 7.98 |
| CHEMBL254219 | DIGITOXIN | 4.0 | 1 | 7.96 |
| CHEMBL107 | COLCHICINE | 4.0 | 1 | 7.95 |
| CHEMBL451887 | CARFILZOMIB | 4.0 | 1 | 7.69 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | 4.0 | 1 | 7.68 |
| CHEMBL917 | FLOXURIDINE | 4.0 | 1 | 7.67 |
| CHEMBL2355712 | — | — | 1 | 7.59 |
| CHEMBL429023 | ROTENONE | — | 1 | 7.59 |
| CHEMBL359744 | DOXORUBICIN HYDROCHLORIDE | 4.0 | 1 | 7.37 |
| CHEMBL1200485 | SORAFENIB TOSYLATE | 4.0 | 1 | 7.33 |
| CHEMBL477772 | PAZOPANIB | 4.0 | 1 | 7.33 |
| CHEMBL167731 | PIXANTRONE | 4.0 | 1 | 7.33 |
| CHEMBL528271 | PARBENDAZOLE | 2.0 | 1 | 7.28 |
| CHEMBL1545634 | — | — | 1 | 7.22 |
| CHEMBL1614 | DESLANOSIDE | 4.0 | 1 | 7.21 |
| CHEMBL110309 | — | — | 1 | 7.15 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | 4.0 | 1 | 7.05 |
| CHEMBL1320139 | HELIOMYCIN | 2.0 | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1554 | DACTINOMYCIN | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL113051 | GIMATECAN | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 2.3 | nM | 8.64 |
| CHEMBL378544 | VINBLASTINE SULFATE | IC50 | = | 2.6 | nM | 8.59 |
| CHEMBL3182961 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3559830 | — | IC50 | = | 4.1 | nM | 8.39 |
| CHEMBL1417019 | MITOXANTRONE HYDROCHLORIDE | IC50 | = | 4.4 | nM | 8.36 |
| CHEMBL538943 | VINORELBINE TARTRATE | IC50 | = | 5.5 | nM | 8.26 |
| CHEMBL2354444 | PIRARUBICIN | IC50 | = | 6.3 | nM | 8.20 |
| CHEMBL90555 | VINCRISTINE | IC50 | = | 6.5 | nM | 8.19 |
| CHEMBL61 | PODOFILOX | IC50 | = | 8.1 | nM | 8.09 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | IC50 | = | 10.5 | nM | 7.98 |
| CHEMBL254219 | DIGITOXIN | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL107 | COLCHICINE | IC50 | = | 11.2 | nM | 7.95 |
| CHEMBL451887 | CARFILZOMIB | IC50 | = | 20.4 | nM | 7.69 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | IC50 | = | 20.8 | nM | 7.68 |
| CHEMBL917 | FLOXURIDINE | IC50 | = | 21.6 | nM | 7.67 |
| CHEMBL429023 | ROTENONE | IC50 | = | 25.7 | nM | 7.59 |
| CHEMBL2355712 | — | IC50 | = | 25.4 | nM | 7.59 |
| CHEMBL359744 | DOXORUBICIN HYDROCHLORIDE | IC50 | = | 42.9 | nM | 7.37 |
| CHEMBL167731 | PIXANTRONE | IC50 | = | 46.5 | nM | 7.33 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 46.5 | nM | 7.33 |
| CHEMBL1200485 | SORAFENIB TOSYLATE | IC50 | = | 46.8 | nM | 7.33 |
| CHEMBL528271 | PARBENDAZOLE | IC50 | = | 53.0 | nM | 7.28 |
| CHEMBL1545634 | — | IC50 | = | 60.5 | nM | 7.22 |
| CHEMBL1614 | DESLANOSIDE | IC50 | = | 61.4 | nM | 7.21 |
| CHEMBL110309 | — | IC50 | = | 70.2 | nM | 7.15 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | IC50 | = | 89.4 | nM | 7.05 |
| CHEMBL1320139 | HELIOMYCIN | IC50 | = | 100.5 | nM | 7.00 |
| CHEMBL9514 | NOCODAZOLE | IC50 | = | 101.8 | nM | 6.99 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 101.9 | nM | 6.99 |
| CHEMBL3184888 | — | IC50 | = | 109.1 | nM | 6.96 |
| CHEMBL101253 | VATALANIB | IC50 | = | 110.9 | nM | 6.96 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 112.0 | nM | 6.95 |
| CHEMBL2105698 | ALVOCIDIB HYDROCHLORIDE | IC50 | = | 113.8 | nM | 6.94 |
| CHEMBL3561919 | — | IC50 | = | 154.6 | nM | 6.81 |
| CHEMBL64894 | GENTIAN VIOLET | IC50 | = | 185.9 | nM | 6.73 |
| CHEMBL37161 | FENBENDAZOLE | IC50 | = | 206.7 | nM | 6.68 |
| CHEMBL2356502 | — | IC50 | = | 251.7 | nM | 6.60 |
| CHEMBL42442 | OXFENDAZOLE | IC50 | = | 288.4 | nM | 6.54 |
| CHEMBL1087630 | OXIBENDAZOLE | IC50 | = | 327.6 | nM | 6.49 |
| CHEMBL1483 | ALBENDAZOLE | IC50 | = | 355.4 | nM | 6.45 |
| CHEMBL140144 | — | IC50 | = | 354.4 | nM | 6.45 |
| CHEMBL685 | MEBENDAZOLE | IC50 | = | 369.9 | nM | 6.43 |
| CHEMBL105442 | CI-1040 | IC50 | = | 368.4 | nM | 6.43 |
| CHEMBL31907 | CETABEN | IC50 | = | 367.3 | nM | 6.43 |
| CHEMBL922 | ADEFOVIR DIPIVOXIL | IC50 | = | 391.3 | nM | 6.41 |
| CHEMBL554041 | ALEXIDINE DIHYDROCHLORIDE | IC50 | = | 407.8 | nM | 6.39 |