Assay Detail
Functional
CHEMBL3562060
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Dose response counterscreen for inhibitors of viability of late stage Plasmodium falciparum gametocytes: Luminescence-based cell-based high throughput dose response assay to identify compounds that are cytotoxic to Jurkat human T lymphocyte cells.. (Class of assay: confirmatory)
244
Total Activities
244
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | Jurkat |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 244 | 4.75 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL560906 | — | — | 1 | 6.46 |
| CHEMBL1488923 | — | — | 1 | 5.62 |
| CHEMBL1612044 | — | — | 1 | 5.40 |
| CHEMBL1310318 | — | — | 1 | 5.17 |
| CHEMBL1562606 | — | — | 1 | 5.16 |
| CHEMBL1422167 | — | — | 1 | 4.96 |
| CHEMBL1532997 | — | — | 1 | 4.65 |
| CHEMBL1497135 | — | — | 1 | 4.45 |
| CHEMBL1725121 | — | — | 1 | 4.42 |
| CHEMBL1425183 | — | — | 1 | 4.36 |
| CHEMBL1370269 | — | — | 1 | 4.19 |
| CHEMBL1372869 | — | — | 1 | 4.16 |
| CHEMBL1510254 | — | — | 1 | 4.12 |
| CHEMBL1344417 | — | — | 1 | 4.10 |
| CHEMBL1501983 | — | — | 1 | 4.09 |
| CHEMBL1577914 | — | — | 1 | - |
| CHEMBL1735080 | — | — | 1 | - |
| CHEMBL1341808 | — | — | 1 | - |
| CHEMBL1901165 | — | — | 1 | - |
| CHEMBL1390245 | — | — | 1 | - |
| CHEMBL2141346 | — | — | 1 | - |
| CHEMBL1471955 | — | — | 1 | - |
| CHEMBL1374100 | — | — | 1 | - |
| CHEMBL1450241 | — | — | 1 | - |
| CHEMBL1450769 | — | — | 1 | - |
| CHEMBL1306159 | — | — | 1 | - |
| CHEMBL1371320 | — | — | 1 | - |
| CHEMBL1392521 | — | — | 1 | - |
| CHEMBL1499751 | — | — | 1 | - |
| CHEMBL1299736 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL560906 | — | IC50 | = | 349.74 | nM | 6.46 |
| CHEMBL1488923 | — | IC50 | = | 2413.0 | nM | 5.62 |
| CHEMBL1612044 | — | IC50 | = | 3976.0 | nM | 5.40 |
| CHEMBL1310318 | — | IC50 | = | 6728.0 | nM | 5.17 |
| CHEMBL1562606 | — | IC50 | = | 6869.0 | nM | 5.16 |
| CHEMBL1422167 | — | IC50 | = | 10923.0 | nM | 4.96 |
| CHEMBL1532997 | — | IC50 | = | 22217.0 | nM | 4.65 |
| CHEMBL1497135 | — | IC50 | = | 35598.0 | nM | 4.45 |
| CHEMBL1725121 | — | IC50 | = | 37798.0 | nM | 4.42 |
| CHEMBL1425183 | — | IC50 | = | 43566.0 | nM | 4.36 |
| CHEMBL1370269 | — | IC50 | = | 64418.0 | nM | 4.19 |
| CHEMBL1372869 | — | IC50 | = | 68604.0 | nM | 4.16 |
| CHEMBL1510254 | — | IC50 | = | 76192.0 | nM | 4.12 |
| CHEMBL1344417 | — | IC50 | = | 79253.0 | nM | 4.10 |
| CHEMBL1501983 | — | IC50 | = | 80619.0 | nM | 4.09 |
| CHEMBL3561308 | — | IC50 | > | 83271.0 | nM | - |
| CHEMBL2132231 | — | IC50 | > | 83325.0 | nM | - |
| CHEMBL1611944 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1891973 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1537115 | — | IC50 | > | 83288.0 | nM | - |
| CHEMBL1488986 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1454182 | — | IC50 | > | 83282.0 | nM | - |
| CHEMBL1370291 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1563978 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1599872 | — | IC50 | > | 83317.0 | nM | - |
| CHEMBL1537854 | — | IC50 | > | 83300.0 | nM | - |
| CHEMBL1584386 | — | IC50 | > | 83239.0 | nM | - |
| CHEMBL1438544 | — | IC50 | > | 83392.0 | nM | - |
| CHEMBL1423114 | — | IC50 | > | 83367.0 | nM | - |
| CHEMBL1309203 | — | IC50 | > | 83295.0 | nM | - |
| CHEMBL1550466 | — | IC50 | > | 83289.0 | nM | - |
| CHEMBL1540629 | — | IC50 | > | 83290.0 | nM | - |
| CHEMBL1904115 | — | IC50 | > | 83317.0 | nM | - |
| CHEMBL1611650 | — | IC50 | > | 83297.0 | nM | - |
| CHEMBL1429875 | — | IC50 | > | 83300.0 | nM | - |
| CHEMBL1377718 | — | IC50 | > | 83292.0 | nM | - |
| CHEMBL1483420 | — | IC50 | > | 83299.0 | nM | - |
| CHEMBL1402896 | — | IC50 | > | 83174.0 | nM | - |
| CHEMBL1428728 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1448921 | — | IC50 | > | 83269.0 | nM | - |
| CHEMBL1732171 | — | IC50 | > | 83334.0 | nM | - |
| CHEMBL1390959 | — | IC50 | > | 83367.0 | nM | - |
| CHEMBL1509711 | — | IC50 | > | 83234.0 | nM | - |
| CHEMBL1351569 | — | IC50 | > | 83272.0 | nM | - |
| CHEMBL1477713 | — | IC50 | > | 83300.0 | nM | - |
| CHEMBL1335486 | — | IC50 | > | 83246.0 | nM | - |
| CHEMBL1426363 | — | IC50 | > | 83359.0 | nM | - |
| CHEMBL1705197 | — | IC50 | > | 83309.0 | nM | - |
| CHEMBL1369541 | — | IC50 | > | 83239.0 | nM | - |
| CHEMBL1402652 | — | IC50 | > | 83325.0 | nM | - |