Assay Detail
Binding
CHEMBL3584796
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Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assay
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | RBE4 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Monocarboxylate transporter 1 (CHEMBL2073709) ↗| Type | SINGLE PROTEIN |
| Organism | Rattus norvegicus |
Publication
Monocarboxylate transporter 1 inhibitors as potential anticancer agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 7.03 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3582422 | — | — | 1 | 8.10 |
| CHEMBL3582419 | — | — | 1 | 8.05 |
| CHEMBL3582408 | — | — | 1 | 8.00 |
| CHEMBL3582423 | — | — | 1 | 7.96 |
| CHEMBL3582420 | — | — | 1 | 7.96 |
| CHEMBL3582418 | — | — | 1 | 7.92 |
| CHEMBL3582426 | — | — | 1 | 7.60 |
| CHEMBL3582424 | — | — | 1 | 7.54 |
| CHEMBL3582409 | — | — | 1 | 7.52 |
| CHEMBL3582415 | — | — | 1 | 7.52 |
| CHEMBL3582421 | — | — | 1 | 7.47 |
| CHEMBL3582425 | — | — | 1 | 7.32 |
| CHEMBL3582407 | — | — | 1 | 7.16 |
| CHEMBL3582416 | — | — | 1 | 7.16 |
| CHEMBL3582410 | — | — | 1 | 7.00 |
| CHEMBL3582413 | — | — | 1 | 6.96 |
| CHEMBL77436 | — | — | 1 | 6.85 |
| CHEMBL3582411 | — | — | 1 | 6.85 |
| CHEMBL3582417 | — | — | 1 | 6.85 |
| CHEMBL3582414 | — | — | 1 | 6.40 |
| CHEMBL3582406 | — | — | 1 | 6.30 |
| CHEMBL77524 | — | — | 1 | 6.30 |
| CHEMBL309866 | — | — | 1 | 6.30 |
| CHEMBL3582405 | — | — | 1 | 6.30 |
| CHEMBL3582404 | — | — | 1 | 6.30 |
| CHEMBL3582403 | — | — | 1 | 6.30 |
| CHEMBL78184 | — | — | 1 | 6.30 |
| CHEMBL3582402 | — | — | 1 | 6.30 |
| CHEMBL77278 | — | — | 1 | 6.30 |
| CHEMBL3582412 | — | — | 1 | 6.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3582422 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL3582419 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL3582408 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL3582423 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL3582420 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL3582418 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL3582426 | — | IC50 | = | 25.0 | nM | 7.60 |
| CHEMBL3582424 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL3582409 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL3582415 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL3582421 | — | IC50 | = | 34.0 | nM | 7.47 |
| CHEMBL3582425 | — | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL3582407 | — | IC50 | = | 70.0 | nM | 7.16 |
| CHEMBL3582416 | — | IC50 | = | 70.0 | nM | 7.16 |
| CHEMBL3582410 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL3582413 | — | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL77436 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL3582411 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL3582417 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL3582414 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL3582406 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL77524 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL309866 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3582405 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3582404 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3582403 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL78184 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3582402 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL77278 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL3582412 | — | IC50 | = | 880.0 | nM | 6.06 |