Assay Detail
Binding
CHEMBL3587785
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Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells by microplate scintillation counting
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.04 | 7.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL80 | NALOXONE | 4.0 | 1 | 7.52 |
| CHEMBL226508 | — | — | 1 | 5.51 |
| CHEMBL78010 | PECTOLINARIGENIN | — | 1 | 5.08 |
| CHEMBL376644 | SALVIGENIN | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL80 | NALOXONE | Ki | = | 30.0 | nM | 7.52 |
| CHEMBL226508 | — | Ki | = | 3100.0 | nM | 5.51 |
| CHEMBL78010 | PECTOLINARIGENIN | Ki | = | 8400.0 | nM | 5.08 |
| CHEMBL376644 | SALVIGENIN | Ki | > | 26000.0 | nM | - |