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Assay Detail

CHEMBL3608048

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to adenosine A2A receptor in rat brain striatal membranes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Tissue Brain
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Adenosine receptor A2a (CHEMBL302)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

New Frontiers in Selective Human MAO-B Inhibitors.
Carradori S, Silvestri R.
J Med Chem (2015) 58 : 6717 -6732
PubMed 25915162 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.44 7.44

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL26138 1 7.44

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL26138 Ki = 36.0 nM 7.44