Assay Detail
Binding
CHEMBL3707633
Review assay metadata, readout intent, target linkage, and publication context from the same page.
ATP Depletion Assay: The activity of PIM1, PIM2, and PIM3 is measured using a luciferase-luciferin based ATP detection reagent to quantify ATP depletion resulting from kinase-catalyzed phosphoryl transfer to a peptide substrate.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Serine/threonine-protein kinase pim-3 (CHEMBL5407) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Kinase inhibitors and methods of their use
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 8.37 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3651899 | — | — | 1 | 9.00 |
| CHEMBL3652019 | — | — | 1 | 9.00 |
| CHEMBL3652008 | — | — | 1 | 9.00 |
| CHEMBL3652022 | — | — | 1 | 9.00 |
| CHEMBL3651994 | — | — | 1 | 9.00 |
| CHEMBL3651920 | — | — | 1 | 9.00 |
| CHEMBL3652010 | — | — | 1 | 9.00 |
| CHEMBL3652006 | — | — | 1 | 9.00 |
| CHEMBL3652004 | — | — | 1 | 9.00 |
| CHEMBL3105022 | — | — | 1 | 9.00 |
| CHEMBL3652018 | — | — | 1 | 9.00 |
| CHEMBL3105021 | — | — | 1 | 9.00 |
| CHEMBL3652009 | — | — | 1 | 9.00 |
| CHEMBL3651947 | — | — | 2 | 9.00 |
| CHEMBL3651953 | — | — | 1 | 8.70 |
| CHEMBL3651945 | — | — | 1 | 8.70 |
| CHEMBL3651962 | — | — | 1 | 8.70 |
| CHEMBL3652015 | — | — | 1 | 8.70 |
| CHEMBL3652016 | — | — | 1 | 8.70 |
| CHEMBL3651924 | — | — | 1 | 8.70 |
| CHEMBL3651921 | — | — | 1 | 8.70 |
| CHEMBL3651948 | — | — | 1 | 8.70 |
| CHEMBL3651923 | — | — | 1 | 8.70 |
| CHEMBL3651941 | — | — | 1 | 8.70 |
| CHEMBL3651955 | — | — | 1 | 8.70 |
| CHEMBL3651940 | — | — | 1 | 8.70 |
| CHEMBL3651981 | — | — | 1 | 8.70 |
| CHEMBL3651904 | — | — | 1 | 8.70 |
| CHEMBL3652011 | — | — | 1 | 8.70 |
| CHEMBL3651942 | — | — | 1 | 8.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3652004 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3105022 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3651994 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3651920 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3651947 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652009 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3651899 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3105021 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652010 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652018 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652006 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652022 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652019 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3652008 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL3651924 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652023 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651966 | LGH-447 | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651959 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652003 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651955 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651903 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651922 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651904 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651972 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651938 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651940 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651942 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651981 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652011 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651905 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651923 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651939 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651936 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651953 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651946 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652013 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651945 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651962 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652015 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652016 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651900 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3652017 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651921 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651948 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651941 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3651963 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3651956 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3651932 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3651916 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL3651912 | — | IC50 | = | 3.0 | nM | 8.52 |